The 5-HT1 receptors are a subfamily of the 5-HT serotonin receptors that bind to the endogenous neurotransmitter serotonin (also known as 5-hydroxytryptamine...
5 KB (472 words) - 15:42, 23 May 2025
serotonin receptor agonist is an agonist of one or more serotonin receptors. They activate serotonin receptors in a manner similar to that of serotonin (5-hydroxytryptamine;...
16 KB (1,664 words) - 07:32, 20 February 2025
5-hydroxytryptamine (serotonin) receptor 1F, also known as HTR1F is a 5-HT1 receptor protein and also denotes the human gene encoding it. 5-n-Butyryloxy-DMT:...
9 KB (1,053 words) - 16:05, 22 May 2025
Chamomile (ethanol extract) 5-HT receptor 5-HT1 receptor 5-HT2 receptor 5-HT3 receptor 5-HT5 receptor 5-HT6 receptor 5-HT7 receptor GRCh38: Ensembl release...
18 KB (2,096 words) - 04:06, 20 May 2025
of receptors were classed as "5-HT1-like" - by 1998 it was being argued that, since these receptors were "a heterogeneous population of 5-HT1B, 5-HT1D...
65 KB (5,273 words) - 08:55, 28 May 2025
of 5-HT3 receptors in cell lines and native tissues quickly followed. 5-HT1 receptor 5-HT2 receptor 5-HT4 receptor 5-HT5 receptor 5-HT6 receptor 5-HT7...
23 KB (2,440 words) - 22:20, 30 May 2025
5-hydroxytryptamine (serotonin) 1E receptor (5-HT1E) is a highly expressed human G-protein coupled receptor that belongs to the 5-HT1 receptor family (Gi-coupled...
9 KB (1,202 words) - 15:59, 22 May 2025
5-HT2A receptor 5-HT2B receptor 5-HT2C receptor 5-HT1 receptor 5-HT3 receptor 5-HT4 receptor 5-HT5 receptor 5-HT6 receptor 5-HT7 receptor Category:5-HT2...
2 KB (166 words) - 00:47, 13 May 2022
Paliperidone Risperidone 5-HT receptor 5-HT1 receptor 5-HT2 receptor 5-HT3 receptor 5-HT4 receptor 5-HT5 receptor 5-HT6 receptor GRCh38: Ensembl release...
26 KB (3,078 words) - 21:46, 20 May 2025
relation to Parkinson's disease. 5-HT receptor 5-HT1 receptor 5-HT2 receptor 5-HT3 receptor 5-HT4 receptor 5-HT5 receptor GRCh38: Ensembl release 89: ENSG00000158748...
29 KB (3,306 words) - 05:19, 25 May 2025
Cyproheptadine blocks 5-HT2A, H1 and is a mild anticholinergic. Methysergide is a 5-HT2A antagonist and nonselective 5-HT1 receptor blocker. It causes retroperitoneal...
5 KB (503 words) - 05:28, 26 March 2025
(antidepressant) GR-127935 (mixed 5-HT1B/1D antagonist) LY-310762 LY-367642 LY-456219 LY-456220 5-HT1 receptor 5-HT receptor GRCh38: Ensembl release 89: ENSG00000179546...
11 KB (1,241 words) - 12:55, 30 May 2025
206 nM affinity. SB-699,551 5-HT receptor 5-HT1 receptor 5-HT2 receptor 5-HT3 receptor 5-HT4 receptor 5-HT6 receptor 5-HT7 receptor GRCh38: Ensembl release...
16 KB (1,773 words) - 06:08, 29 April 2025
with respect to personality traits and showed no major effect. 5-HT1 receptor 5-HT receptor GRCh38: Ensembl release 89: ENSG00000135312 – Ensembl, May 2017...
23 KB (2,513 words) - 10:28, 14 April 2025
receptor (or 5-HT1A receptor) is a subtype of serotonin receptors, or 5-HT receptors, that binds serotonin, also known as 5-HT, a neurotransmitter. 5-HT1A...
59 KB (6,182 words) - 23:06, 22 May 2025
Serotonin (redirect from 5-Hydroxytryptamine)
serotonin receptors, including the serotonin 5-HT1 (1A, 1B, 1D, 1E, 1F), 5-HT2 (2A, 2B, 2C), 5-HT3, 5-HT4, 5-HT5 (5A, 5B), 5-HT6, and 5-HT7 receptors. Except...
173 KB (18,295 words) - 19:45, 2 June 2025
acute MDMA intoxication on mood and impulsivity: role of the 5-HT2 and 5-HT1 receptors". PLOS ONE. 7 (7): e40187. Bibcode:2012PLoSO...740187V. doi:10...
63 KB (6,729 words) - 22:17, 2 June 2025
Rizatriptan (category 5-HT1D agonists)
Rizatriptan is in the triptan class and is believed to work by activating the 5-HT1 receptor. Rizatriptan was patented in 1991 and came into medical use in 1998...
12 KB (686 words) - 12:10, 3 June 2025
was 100 nM in the same study. 3,4-DMA also showed affinity for the 5-HT1 receptor (Ki = 64,600 nM). The drug has additionally been found to be a monoamine...
7 KB (496 words) - 22:53, 17 June 2025
Methysergide (category Serotonin receptor agonists)
agonist of some serotonin receptors (e.g., the 5-HT1 receptors) and antagonist of other serotonin receptors (e.g., the 5-HT2 receptors), methylergonovine is...
32 KB (2,699 words) - 21:25, 18 May 2025
Locomotor activity (section Dopamine receptor agonists)
with chronic administration. The dual TAAR1 full agonist and serotonin 5-HT1 receptor modulator ulotaront did not affect dextroamphetamine-induced hyperlocomotion...
114 KB (12,382 words) - 04:41, 2 June 2025
label two different 5-HT receptors, and neither of them displaced morphine, leading to naming of the 5-HT1, 5-HT2 and 5-HT3 receptors, corresponding to...
131 KB (13,680 words) - 11:36, 9 June 2025
yield arachidonic acid. Receptors that activate this pathway include: A1 receptor D2 receptor α2 adrenergic receptor 5-HT1 receptor PLC may also be activated...
21 KB (1,892 words) - 13:52, 12 June 2025
Naratriptan (category 5-HT1D agonists)
is used for the treatment of migraine headaches. It is a selective 5-HT1 receptor subtype agonist. It was patented in 1987 and approved for medical use...
11 KB (954 words) - 06:05, 26 May 2025
Ergotamine (category Non-hallucinogenic 5-HT2A receptor agonists)
dopamine receptors. It is an agonist of serotonin receptors including the serotonin 5-HT1 and 5-HT2 subtypes. Ergotamine is an agonist of the serotonin 5-HT2B...
24 KB (1,517 words) - 09:37, 9 May 2025
JRT (drug) (category Serotonin receptor modulators)
affinity for the serotonin 5-HT1B or 5-HT3 receptors, whereas the other serotonin 5-HT1 receptors and the serotonin 5-HT4 receptor were not reported. (+)-JRT...
11 KB (833 words) - 07:11, 14 June 2025
Beatrice (drug) (category Serotonin receptor modulators)
receptors. Its affinities (Ki) were 415 nM for the 5-HT2 receptor and 3,870 nM for the 5-HT1 receptor. The affinity of Beatrice for the serotonin 5-HT2...
6 KB (373 words) - 23:07, 17 June 2025
psilocybin, which act as non-selective serotonin receptor agonists including of the serotonin 5-HT1 and 5-HT2 receptors, have shown prosocial and empathy-enhancing...
70 KB (6,753 words) - 20:17, 18 June 2025
The 5-HT2C receptor is a subtype of the 5-HT2 receptor that binds the endogenous neurotransmitter serotonin (5-hydroxytryptamine, 5-HT). Like all 5-HT2...
51 KB (6,133 words) - 17:35, 28 May 2025
5-HT1A receptor full agonist PSIL-001 (DMT analogue) – serotonin 5-HT1 receptor modulator (non-hallucinogenic) PSIL-002 (DMT analogue) – serotonin 5-HT1...
151 KB (11,543 words) - 19:01, 18 June 2025