An antigonadotropin is a drug which suppresses the activity and/or downstream effects of one or both of the gonadotropins, follicle-stimulating hormone...
8 KB (794 words) - 07:50, 29 April 2024
Steroidal antiandrogen (category Antigonadotropins)
Cyproterone acetate (Androcur): A combined AR antagonist and progestogen/antigonadotropin. Also has weak glucocorticoid activity. Previously used widely in the...
24 KB (2,340 words) - 08:04, 7 February 2024
Danazol (category Antigonadotropins)
as a weak androgen and anabolic steroid, a weak progestogen, a weak antigonadotropin, a weak steroidogenesis inhibitor, and a functional antiestrogen. Danazol...
46 KB (3,954 words) - 04:46, 8 April 2024
Antiandrogen (section Antigonadotropins)
and antigonadotropins. AR antagonists work by directly blocking the effects of androgens, while androgen synthesis inhibitors and antigonadotropins work...
158 KB (15,044 words) - 16:15, 8 June 2024
of a polymer's viscoelasticity Delmadinone acetate, a progestin and antigonadotropin used as an antiandrogen Dimethandrolone, an anabolic–androgenic steroid...
2 KB (344 words) - 20:17, 8 November 2023
diet or quack preparations, which are illegal in various countries. Antigonadotropin Gonadotropin surge-attenuating factor Parhar, Ishwar S. (2002)....
11 KB (1,114 words) - 19:59, 4 April 2022
(SERD) fulvestrant, aromatase inhibitors (AIs) like anastrozole, and antigonadotropins including androgens/anabolic steroids, progestogens, and GnRH analogues...
9 KB (803 words) - 11:32, 4 January 2024
Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins D2 receptor antagonists (prolactin releasers) (e.g., domperidone,...
210 KB (21,565 words) - 02:49, 29 May 2024
Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins D2 receptor antagonists (prolactin releasers) (e.g., domperidone,...
187 KB (18,318 words) - 01:32, 24 May 2024
List of antiandrogens (section Antigonadotropins)
inhibitors like 5α-reductase inhibitors and CYP17A1 inhibitors, and antigonadotropins like GnRH analogues, estrogens, and progestogens. In addition, it...
5 KB (254 words) - 18:23, 18 September 2023
Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins D2 receptor antagonists (prolactin releasers) (e.g., domperidone,...
50 KB (4,374 words) - 15:14, 13 May 2024
Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins D2 receptor antagonists (prolactin releasers) (e.g., domperidone,...
67 KB (6,821 words) - 14:50, 18 March 2024
Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins D2 receptor antagonists (prolactin releasers) (e.g., domperidone,...
29 KB (3,165 words) - 22:29, 23 March 2024
Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins D2 receptor antagonists (prolactin releasers) (e.g., domperidone,...
23 KB (1,901 words) - 09:38, 9 June 2024
Estrogen (category Antigonadotropins)
Fadrozole Formestane Third-generation: Anastrozole Exemestane Letrozole Antigonadotropins Androgens/anabolic steroids (e.g., testosterone, testosterone esters...
72 KB (7,575 words) - 12:18, 7 June 2024
Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins D2 receptor antagonists (prolactin releasers) (e.g., domperidone,...
47 KB (4,553 words) - 07:12, 2 May 2024
Desogestrel (category Antigonadotropins)
In addition, desogestrel has been extensively investigated as an antigonadotropin at dosages of 150 to 300 μg/day in combination with testosterone in...
63 KB (5,553 words) - 13:39, 12 June 2024
GnRH agonists (e.g., GnRHTooltip gonadotropin-releasing hormone) Antigonadotropins Sex steroid agonists (via negative feedback on the HPG axis): Androgens/anabolic...
49 KB (5,368 words) - 15:05, 11 June 2024
Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins D2 receptor antagonists (prolactin releasers) (e.g., domperidone,...
150 KB (15,741 words) - 22:02, 27 May 2024
Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins D2 receptor antagonists (prolactin releasers) (e.g., domperidone,...
74 KB (7,440 words) - 21:41, 12 June 2024
GnRH agonists (e.g., GnRHTooltip gonadotropin-releasing hormone) Antigonadotropins Sex steroid agonists (via negative feedback on the HPG axis): Androgens/anabolic...
32 KB (3,477 words) - 20:14, 3 June 2024
precursor of cyproterone acetate (CPA), an antiandrogen, progestin, and antigonadotropin which was introduced instead of cyproterone and is widely used as a...
23 KB (2,373 words) - 22:25, 20 February 2024
testosterone levels; antiandrogens such as androgen receptor antagonists, antigonadotropins, GnRH modulators, and 5α-reductase inhibitors to further oppose the...
233 KB (24,875 words) - 03:35, 27 May 2024
Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins D2 receptor antagonists (prolactin releasers) (e.g., domperidone,...
27 KB (2,274 words) - 02:54, 22 March 2024
a progestogen, antigonadotropin, and antiandrogen. It is 2- to 3-fold as potent as spironolactone as a progestogen and antigonadotropin but its antiandrogenic...
6 KB (371 words) - 13:11, 24 December 2023
Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins D2 receptor antagonists (prolactin releasers) (e.g., domperidone,...
7 KB (542 words) - 21:26, 19 February 2024
Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins D2 receptor antagonists (prolactin releasers) (e.g., domperidone,...
23 KB (2,061 words) - 17:44, 8 March 2024
Fadrozole Formestane Third-generation: Anastrozole Exemestane Letrozole Antigonadotropins Androgens/anabolic steroids (e.g., testosterone, testosterone esters...
44 KB (4,550 words) - 01:52, 6 May 2024
Fezolinetant (category Antigonadotropins)
Fezolinetant, sold under the brand name Veozah among others, is a medication used for the treatment of hot flashes (vasomotor symptoms) due to menopause...
17 KB (1,279 words) - 05:53, 10 June 2024
Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins D2 receptor antagonists (prolactin releasers) (e.g., domperidone,...
92 KB (9,319 words) - 21:15, 8 June 2024