A channel modulator, or ion channel modulator, is a type of drug which modulates ion channels. They include channel blockers and channel openers. Ion channels...

3 possibilities). This yields 17 possible modulator combinations. There are 18 (=2*3*3) if neutral modulator type is also included. For all practical considerations...

An RF modulator (radio frequency modulator) is an electronic device used to convert signals from devices such as media players, VCRs and game consoles...

hemopressin, drugs to treat obesity, and more besides. Channel modulator Transporter modulator van Westen GJ, Gaulton A, Overington JP (April 2014). "Chemical...

Chloride channel openers refer to a specific category of drugs designed to modulate chloride channels in the human body. Chloride channels are anion-selective...

A release modulator, or neurotransmitter release modulator, is a type of drug that modulates the release of one or more neurotransmitters. Examples of...

A reuptake modulator, or transporter modulator, is a type of drug which modulates the reuptake of one or more neurotransmitters via their respective neurotransmitter...

Calcium channel blockers (CCB), calcium channel antagonists or calcium antagonists are a group of medications that disrupt the movement of calcium (Ca2+)...

Sodium channel blockers are drugs which impair the conduction of sodium ions (Na+) through sodium channels. The following naturally-produced substances...

the real-valued modulated physical signal (the so-called passband signal or RF signal). These are the general steps used by the modulator to transmit data:...

Development and discovery of SSRI drugs Channel modulator, for links to articles referring to drugs that modulate ion channels. List of monoclonal antibodies List...

Capsicum plants are dispersed predominantly by birds. In birds, the TRPV1 channel does not respond to capsaicin or related chemicals, but mammalian TRPV1...

bees, sea snails, and others) work by modulating ion channel conductance and/or kinetics. In addition, ion channels are key components in a wide variety...

sensation of pain. In addition to regulating channel gating, sodium channel beta subunits also modulate channel expression and form links to the intracellular...

receptor modulator Cannabidivarin (CBDV; GWP-42006) – cannabinoid receptor modulator CMX-020 – TRPV1 modulator as well as CB1 and CB2 receptor modulator Dronabinol...

sodium channel modulator—is also approved for the treatment of moderate to severe pain in some countries. Flupirtine is a centrally acting K+ channel opener...

v t e TRP channel modulators TRPA TRPC TRPM TRPML TRPP TRPV See also: Receptor/signaling modulators • Ion channel modulators...

studies show that menthol acts as a GABAA receptor positive allosteric modulator and increases GABAergic transmission in PAG neurons. Menthol has anesthetic...

of pharmacological modulators of potassium channels, see potassium channel blocker and potassium channel opener. Potassium channels have a tetrameric structure...

Inhibitor ♦ Ion channel: Opener Blocker ♦ Receptor: Agonist Partial agonist Antagonist Inverse agonist Positive allosteric modulator (PAM) Negative allosteric...

positive allosteric modulator Cannabidiol (CBD; GW-42003, GWP-42003, GWP-42003-P, ECP-012A; Arvisol, Epidiolex) – cannabinoid receptor modulator, antioxidant...

standards dictate that CH2 is a 6 MHz wide channel with its luminance carrier at 55.25 MHz, so the modulator for channel 2 will impose the appropriate input...

caused by release of catecholamines. The venom also contains a sodium channel modulator. The sting is moderately irritating; the severe syndrome is delayed...

channels (big potassium), are large conductance calcium-activated potassium channels, and is also known as BKCa, Maxi-K, slo1, or Kca1.1. BK channels...

Foadi N, et al. (2009). "The nonpsychotropic cannabinoid cannabidiol modulates and directly activates alpha-1 and alpha-1-Beta glycine receptor function"...

Voltage-gated sodium channels (VGSCs), also known as voltage-dependent sodium channels (VDSCs), are a group of voltage-gated ion channels found in the membrane...

selectively inhibited Nav1.8 channels, but not other voltage-gated sodium channels, and bound to a unique site on these sodium channels with a novel allosteric...

co-expressed with β subunits. The β subunit acts as an important modulator of channel electrophysiological properties. Until very recently, the interaction...

associated with exposure to tear gas often require medical attention. TRPA1 ion channels expressed on nociceptors have been implicated as the site of action for...

an RF modulator that generates the proper carrier (often for channel 3 or 4 in North America, channel 36 in Europe). Sometimes this modulator is built...