An enzyme inducer is a type of drug that increases the metabolic activity of an enzyme either by binding to the enzyme and activating it, or by increasing...

Enzyme catalysis is the increase in the rate of a process by an "enzyme", a biological molecule. Most enzymes are proteins, and most such processes are...

An adaptive enzyme or inducible enzyme is an enzyme that is expressed only under conditions in which it is clearly of adaptive value, as opposed to a...

secretion, promoting glucose uptake storing it as glycogen in the muscles. Enzyme inducer Effector (biology) Chen G, Zhang Y, Liang J, Li W, Zhu Y, Zhang M, Wang...

In molecular biology, an inducer is a molecule that regulates gene expression. An inducer functions in two ways; namely: By disabling repressors. The gene...

(together with André Lwoff). Aryl hydrocarbon receptor Index inducer or just inducer predictably induce metabolism via a given pathway and are commonly used in...

An enzyme (/ˈɛnzaɪm/) is a protein that acts as a biological catalyst by accelerating chemical reactions. The molecules upon which enzymes may act are...

An enzyme repressor is a type of regulatory protein that controls the activity of enzymes, typically by binding to specific sites on DNA or directly to...

sacred plant and used as an entheogen. Its roots are traditionally used to induce vivid (and according to the Xhosa, prophetic) lucid dreams during the initiation...

the muscarinic receptor, for example pilocarpine, or by inhibiting the enzyme acetylcholinesterase, which hydrolyses the acetylcholine in the synapse...

Typically it includes pharmacological agonists and antagonists, but also enzyme inhibitors (such as monoamine oxidase inhibitors). The origins of clinical...

antihistamines utilized for this purpose include hydroxyzine, promethazine (enzyme induction especially helps with codeine and similar prodrug opioids), phenyltoloxamine...

medications described below. All drugs that fall within the class of enzyme inducers increase the clearance and decrease the half-life of methylprednisolone...

contraceptive effectiveness could be lowered, despite lamotrigine not being an enzyme inducer. An assessment of risks versus benefits of CHC is recommended in women...

sulfamethoxazole) also cause Gram-negative bacteria to form spheroplasts. The enzyme lysozyme causes Gram-negative bacteria to form spheroplasts, but only if...

a known enzyme inducer, has decreased the concentration/dose ratio of olanzapine by 33% compared to olanzapine alone. Another enzyme inducer, ritonavir...

transport protein is phosphorylated by a particular protein kinase, which is an enzyme that adds a phosphate group to proteins. The primary function of most neurotransmitter...

drugs include agonists, antagonists, modulators, reuptake inhibitors and enzymes. Adenosinergic Adrenergic Cannabinoidergic Cholinergic Dopaminergic Glutamatergic...

the inducer, either allolactose or IPTG, to the repressor affects the distribution of repressor between the two shapes. Thus, repressor with inducer bound...

the highest degree of hepatic-enzyme induction on record. In addition to being an inducer of CYP3A4, it is also an inducer of CYP1A2, which causes it to...

GABA receptors, they bind to an allosteric site on the receptor and cannot induce a response from the neuron without an actual agonist being present. Drugs...

activation of α1 stimulates the membrane bound enzyme phospholipase C, and activation of α2 inhibits the enzyme adenylate cyclase. Inactivation of adenylate...

strong enzyme-inducing ASMs. The effect of weak enzyme-inducing ASMs on hormonal contraception is less clear than that of the strong enzyme-inducing ASMs...

wide variety of mechanisms.[citation needed] Some allosteric modulators induce a conformational change in their target receptor which increases the binding...

expresses the higher affinity. The activation of β1, β2 and β3 activates the enzyme, adenylate cyclase. This, in turn, leads to the activation of the secondary...

inhibitor of the P450 enzymes CYP1A2, CYP2C9, CYP2C19, CYP2D6, CYP2E1, CYP3A4. By reducing the metabolism of drugs through these enzymes, cimetidine may increase...

in general, both a decrease in slope and a reduced maximum are obtained. Enzyme inhibitor Growth factor receptor inhibitor Selective receptor modulator...

Kabulov S (1992). "[The advantages of benzonal as an inducer of the liver mono-oxygenase enzyme system compared to phenobarbital]". Eksperimental'naia...

impact on each specific enzyme span a broad range, with phenobarbital and secobarbital being the most potent enzyme inducers and butalbital and talbutal...

neurotransmitter in question leaves them vulnerable to degradation via enzymes such as monoamine oxidase (MAO) that exist in the cytoplasm. With vesicular...