The progesterone receptor (PR), also known as NR3C3 or nuclear receptor subfamily 3, group C, member 3, is a protein found inside cells. It is activated...
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The progesterone receptor C (PR-C) is one of three known isoforms of the progesterone receptor (PR), the main biological target of the endogenous progestogen...
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prescribed in 1934. Progesterone is the most important progestogen in the body. As a potent agonist of the nuclear progesterone receptor (nPR) (with an affinity...
124 KB (11,630 words) - 10:40, 20 May 2025
A selective progesterone receptor modulator (SPRM) is an agent that acts on the progesterone receptor (PR), the biological target of progestogens like...
47 KB (5,150 words) - 21:22, 21 November 2024
The progesterone receptor A (PR-A) is one of three known isoforms of the progesterone receptor (PR), the main biological target of the endogenous progestogen...
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Antiprogestogen (redirect from Progesterone receptor antagonist)
drugs competitively inhibit progestin at progesterone receptors, acting by blocking the progesterone receptor (PR) and/or inhibiting or suppressing progestogen...
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Membrane progesterone receptors (mPRs) are a group of cell surface receptors and membrane steroid receptors belonging to the progestin and adipoQ receptor (PAQR)...
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PRC (disambiguation) (redirect from PrC)
for absorbing light in photosynthesis Progesterone receptor C, one of the isoforms of the progesterone receptor PRC (Palm OS), computer code database...
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hence is an agonist of the progesterone receptor (PR), the biological target of progestogens like endogenous progesterone. It opposes the effects of estrogens...
187 KB (18,628 words) - 21:58, 29 May 2025
receptor (MR; NR3C2) (Aldosterone) 3: Progesterone receptor (PR; NR3C3, PGR) (Sex hormones: Progesterone) 4: Androgen receptor (AR; NR3C4, AR) (Sex hormones:...
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of administration. Progesterone is a naturally occurring and bioidentical progestogen, or an agonist of the progesterone receptor, the biological target...
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– oral progesterone receptor agonist (progestogen/progestin) for prevention of preterm labor VOLT-02 – water-soluble conjugate of progesterone and neurosteroid...
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hormone progesterone. The other isoforms of the PR include the PR-A and PR-C. Membrane progesterone receptor Jacobsen BM, Horwitz KB (2012). "Progesterone receptors...
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The androgen receptor is most closely related to the progesterone receptor, and progestins in higher dosages can block the androgen receptor. The main function...
88 KB (9,471 words) - 05:17, 30 December 2024
The mineralocorticoid receptor (or MR, MLR, MCR), also known as the aldosterone receptor or nuclear receptor subfamily 3, group C, member 2, (NR3C2) is...
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orientated at a 60° angle below the rings C and D. This configuration is ideal for interaction with the progesterone receptor, with retroprogesterone binding with...
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National Laboratory, whose work in isolating and characterizing the progesterone receptor gene has stimulated advances in breast biology and oncology. She...
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Allopregnanolone (category GABAA receptor positive allosteric modulators)
kainate, and glycine receptors. Unlike progesterone, allopregnanolone is inactive at the classical nuclear progesterone receptor (PR). However, allopregnanolone...
51 KB (4,779 words) - 19:54, 29 May 2025
A mineralocorticoid receptor antagonist (MRA or MCRA) or aldosterone antagonist, is a diuretic drug which antagonizes the action of aldosterone at mineralocorticoid...
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or an agonist of the progesterone receptor, the biological target of progestogens like endogenous progesterone. Progesterone also has antimineralocorticoid...
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PGRMC1 (redirect from Progesterone receptor membrane component 1)
Progesterone receptor membrane component 1 (abbreviated PGRMC1) is a protein which co-purifies with progesterone binding proteins in the liver and ovary...
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to estrogen receptor positive tumors (i.e. tumors that contain estrogen receptor positive cells), but can also include progesterone receptor positive tumors...
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progestogen, and hence is an agonist of the progesterone receptor, the biological target of progestogens like progesterone. The medication is an atypical progestogen...
61 KB (6,716 words) - 21:19, 6 January 2025
synthetic steroid hormones that bind to and activate the progesterone receptors (PR). Progesterone is the major and most important progestogen in the body...
16 KB (1,567 words) - 01:04, 8 October 2024
Ulipristal acetate (category Selective progesterone receptor modulators)
is in the selective progesterone receptor modulator (SPRM) class of medications. It works by preventing the effects of progesterone, therefore preventing...
31 KB (2,752 words) - 04:05, 7 March 2025
nuclear receptors include members of subfamily 3, such as the androgen receptor, estrogen receptors, glucocorticoid receptor, and progesterone receptor. It...
75 KB (6,515 words) - 04:42, 1 May 2025
estradiol, estrone, and estriol Progesterone receptor (PR) (A, B) - binds and is activated by progestogens such as progesterone In addition, sex steroids have...
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Hydroxyprogesterone caproate (redirect from 17-alpha-Hydroxy-progesterone caproate)
progestogen, and hence is an agonist of the progesterone receptor, the biological target of progestogens like progesterone. It has some antimineralocorticoid activity...
121 KB (12,026 words) - 21:07, 29 May 2025
Medroxyprogesterone (redirect from Medroxy-progesterone)
(September 2006). "Determination of conformational changes in the progesterone receptor using ELISA-like assays". Steroids. 71 (9): 792–8. doi:10.1016/j...
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among the highest known affinity of any AAS for the androgen (and progesterone) receptors, and has been said to be perhaps the most potent AAS to have ever...
9 KB (511 words) - 06:23, 14 January 2025