The PyrR binding site is an RNA element that is found upstream of a variety of genes involved in pyrimidine biosynthesis and transport. The RNA structure...
2 KB (103 words) - 03:41, 4 October 2019
List of cis-regulatory RNA elements (section R)
Pseudomon-groES RNA motif Pseudomonas rnk leader Pseudomonas rpsL leader PyrG leader PyrR binding site R2 RNA element RbcL 5′ UTR RNA stabilising element Red clover...
6 KB (711 words) - 21:32, 6 October 2024
Index of molecular biology articles (section R)
beta-glucan-transporting ATPase - beta2-adaptin C-terminal domain - binding site - biological organisation - biological process - Biomolecular gradient...
23 KB (1,969 words) - 13:07, 28 September 2024
Giemsa stain (redirect from Giemsa binding)
stain Microscopy Romanowsky stain Wright's stain Zipfel, E.; Grezes, J. -R.; Naujok, A.; Seiffert, W.; Wittekind, D. H.; Zimmermann, H. W. (1984). "Über...
6 KB (619 words) - 02:59, 25 May 2025
List of methylphenidate analogues (section Receptor binding profiles of selected methylphenidate analogues)
measure of fivefold (5×) discrepancy in the entropy of binding at their presumed shared target binding site, which may account for the higher abuse potential...
60 KB (2,336 words) - 17:12, 30 April 2025
5-MeO-pyr-T, also known as 5-methoxy-N,N-tetramethylenetryptamine or as 5-methoxy-3-(2-pyrrolidinoethyl)indole, is a serotonin receptor modulator and...
18 KB (1,700 words) - 03:07, 16 June 2025
(December 2011). "Trace amine-associated receptor 1 is a stereoselective binding site for compounds in the amphetamine class". Bioorg Med Chem. 19 (23): 7044–7048...
31 KB (2,631 words) - 05:37, 10 May 2025
it is hypothesized that AMPT competes with tyrosine at the tyrosine-binding site, causing inhibition of tyrosine hydroxylase. It has been used in the...
25 KB (2,271 words) - 22:29, 15 July 2025
high-affinity, extracellular, and allosteric Zn2+ (zinc ion) binding site which, upon zinc binding, inhibits dopamine reuptake, inhibits amphetamine-induced...
320 KB (34,225 words) - 04:17, 22 July 2025
funnel that is suggested to serve as the insertion site for ubiquinone, in conjunction with the FMN binding cavity at the C-terminal. The two terminal domains...
13 KB (1,324 words) - 03:45, 3 February 2025
given during migraine attacks decreases brain serotonin 5-HT1B receptor binding in humans, with a corresponding receptor occupancy of 16%. However, this...
46 KB (3,880 words) - 19:29, 23 July 2025
Adderall (redirect from Adderall(r))
transporter contains a high affinity extracellular zinc binding site which, upon zinc binding, inhibits dopamine reuptake and amplifies amphetamine-induced...
63 KB (23,111 words) - 16:15, 16 July 2025
receptor indicates binding site structure". Medicinal Chemistry Research. 3: 52–66. Shahar O, Botvinnik A, Esh-Zuntz N, Brownstien M, Wolf R, Lotan A, et al...
268 KB (27,308 words) - 14:15, 18 July 2025
steric interactions between the ring structure and the binding site. Nichols DE, Snyder SE, Oberlender R, Johnson MP, Huang XM (January 1991). "2,3-Dihydrobenzofuran...
13 KB (1,358 words) - 04:08, 14 July 2025
Table II. Affinities of Selected Phenalkylamines for 5-HT1 and 5-HT2 Binding Sites Cerletti A, Taeschler M, Weidmann H (1968). Pharmacologic studies on...
16 KB (1,403 words) - 00:15, 18 June 2025
of non-binding sites on the DAT molecule to exert its own binding, as well as the potential of augmented affinity for NET if its binding site is otherwise...
149 KB (13,608 words) - 22:00, 23 July 2025
family. It is a benzodiazepine site agonist selective for certain subunits. TCS 1205 acts at the benzodiazepine binding site, it is selective for the α1...
3 KB (150 words) - 07:19, 22 June 2025
Phenalkylamines for 5-HT1 and 5-HT2 Binding Sites [...] Shannon M, Battaglia G, Glennon RA, Titeler M (June 1984). "5-HT1 and 5-HT2 binding properties of derivatives...
7 KB (505 words) - 04:57, 19 July 2025
concentrations of 50-100 μmol/L. Its efficacies at the other receptor binding sites are unclear. It has also been shown in vitro to be a substrate for the...
176 KB (17,031 words) - 09:57, 18 July 2025
tryptamine Tetrahydropyridinylindole VU6067416 RS134-49 (R)-69 RU-24,969 EMD-386088 SN-22 MPMI Pyr-T Pip-T Kitson SL (2007). "5-hydroxytryptamine (5-HT)...
7 KB (506 words) - 05:06, 16 July 2025
ibogaine and its principal metabolite (12-hydroxyibogamine) at the MK-801 binding site of the NMDA receptor complex". Neurosci Lett. 192 (1): 53–56. doi:10...
92 KB (8,683 words) - 17:12, 21 July 2025
Urease (section Active site)
the active site cavity when the mobile ‘flap’ (which allows for the entrance of urea into the active site) is open. Stability of the binding of urea to...
36 KB (4,283 words) - 09:14, 5 July 2025
the chemical structure of the site of binding (sulfhydryl, phosphinyl, carboxyl) to the active center of ACE. Kumar R, Chaudhary K, Sharma M, Nagpal...
66 KB (7,220 words) - 01:57, 19 July 2025
of the trimethylsilyl group in 1S-LSD is thought to slightly alter its binding affinity and metabolic profile, although empirical data is still needed...
7 KB (678 words) - 08:41, 20 July 2025
Phenalkylamines for 5-HT1 and 5-HT2 Binding Sites Shannon M, Battaglia G, Glennon RA, Titeler M (June 1984). "5-HT1 and 5-HT2 binding properties of derivatives...
22 KB (1,503 words) - 05:27, 15 July 2025
Phenalkylamines for 5-HT1 and 5-HT2 Binding Sites Shannon M, Battaglia G, Glennon RA, Titeler M (June 1984). "5-HT1 and 5-HT2 binding properties of derivatives...
20 KB (1,189 words) - 23:49, 4 July 2025
reported to have an IC50 of about 50 nM for the inhibition of [3H]5-HT binding, which is at least 5 times less potent than typical reported values for...
7 KB (642 words) - 23:30, 7 July 2025
Erasmus University Repository. Retrieved 19 June 2025. Table 1.2 Receptor binding properties (pKi values) of sumatriptan and second-generation triptans at...
21 KB (1,568 words) - 21:56, 19 July 2025
5-HT2C binding of phenylalkyl- and indolylalkylamines". Journal of Medicinal Chemistry. 37 (13): 1929–35. doi:10.1021/jm00039a004. PMID 8027974. Heim R (March...
55 KB (5,168 words) - 18:39, 16 July 2025
"Angiotensin-Converting Enzyme 2 Metabolizes and Partially Inactivates Pyr-Apelin-13 and Apelin-17: Physiological Effects in the Cardiovascular System"...
24 KB (2,562 words) - 19:53, 23 June 2025