Selective androgen receptor modulators (SARMs) are a class of drugs that selectively activate the androgen receptor in specific tissues, promoting muscle...
74 KB (6,714 words) - 19:02, 22 May 2025
of selective estrogen receptor modulators Selective androgen receptor modulator Selective estrogen receptor degrader Selective receptor modulator Timeline...
58 KB (6,598 words) - 18:11, 25 May 2025
Selective glucocorticoid receptor agonists. Selective receptor modulator Selective androgen receptor modulator Selective estrogen receptor modulator Selective...
25 KB (2,563 words) - 12:23, 11 June 2025
Vosilasarm (category Selective androgen receptor modulators)
and by the black-market name Testolone or Testalone, is a selective androgen receptor modulator (SARM) which is under development for the treatment of hormone-sensitive...
28 KB (2,531 words) - 03:20, 26 May 2025
Enobosarm (category Selective androgen receptor modulators)
MK-2866, and S-22, is a selective androgen receptor modulator (SARM) which is under development for the treatment of androgen receptor-positive breast cancer...
117 KB (12,953 words) - 20:44, 29 May 2025
Antiandrogen (redirect from Androgen receptor antagonist)
for instance androgens and anabolic steroids (AAS) like testosterone, DHT, and nandrolone and selective androgen receptor modulators (SARMs) like enobosarm...
161 KB (15,261 words) - 19:58, 29 May 2025
YK-11 (category Selective androgen receptor modulators)
YK-11 is a synthetic, steroidal selective androgen receptor modulator (SARM) structurally derived from dihydrotestosterone (DHT). It is currently classified...
4 KB (395 words) - 02:19, 1 June 2025
Ligandrol (category Selective androgen receptor modulators)
name VK5211 and by the black-market name Ligandrol, is a selective androgen receptor modulator (SARM) which is under development for the treatment of muscle...
55 KB (6,004 words) - 06:50, 2 June 2025
A selective progesterone receptor modulator (SPRM) is an agent that acts on the progesterone receptor (PR), the biological target of progestogens like...
47 KB (5,156 words) - 23:57, 6 June 2025
allosteric modulators, Examples of receptor modulators in modern medicine include CFTR modulators, selective androgen receptor modulators (SARMs), and...
8 KB (980 words) - 06:37, 28 April 2025
The androgen receptor (AR), also known as NR3C4 (nuclear receptor subfamily 3, group C, member 4), is a type of nuclear receptor that is activated by binding...
88 KB (9,474 words) - 07:42, 9 June 2025
Nonsteroidal antiandrogen (redirect from Nonsteroidal androgen receptor antagonist)
are typically selective and full or silent antagonists of the androgen receptor (AR) and act by directly blocking the effects of androgens like testosterone...
17 KB (1,576 words) - 06:25, 25 May 2025
Andarine (category Selective androgen receptor modulators)
Andarine (developmental code names GTx-007, S-4) is a selective androgen receptor modulator (SARM) which was developed by GTX, Inc for the treatment of...
10 KB (960 words) - 03:05, 14 November 2024
Membrane androgen receptors (mARs) are a group of G protein-coupled receptors (GPCRs), which bind and are activated by testosterone and/or other androgens. Unlike...
5 KB (486 words) - 09:37, 28 February 2025
Classes of selective receptor modulators include: Selective androgen receptor modulator (SARM) Selective estrogen receptor modulator (SERM) Selective glucocorticoid...
2 KB (159 words) - 21:17, 25 March 2025
Anabolic steroid (redirect from Artificial androgen)
and androgens have been found to increase abdominal fat in postmenopausal women and transgender men as well. Selective androgen receptor modulator Antiandrogen...
209 KB (21,562 words) - 04:12, 10 June 2025
A (selective) androgen receptor degrader or downregulator (SARD) is a type of drug which interacts with the androgen receptor (AR) such that it causes...
4 KB (339 words) - 18:32, 17 November 2024
Mostaghel EA, Nelson PS (2021). "Selective androgen receptor modulators activate the canonical prostate cancer androgen receptor program and repress cancer...
35 KB (4,222 words) - 22:11, 19 June 2025
This article pertains to steroidal androgens; nonsteroidal androgens like the selective androgen receptor modulators (SARMs) andarine and enobosarm (ostarine)...
31 KB (754 words) - 23:16, 5 April 2025
Marieta (February 2023). "Exploring the polymorphism of selective androgen receptor modulator YK11". Journal of Molecular Structure. 1273: 134281....
11 KB (1,192 words) - 15:44, 23 May 2025
S-23 (drug) (category Selective androgen receptor modulators)
investigational selective androgen receptor modulator (SARM) developed by GTX, Inc as a potential male hormonal contraceptive. It binds to the androgen receptor more...
3 KB (173 words) - 19:04, 7 January 2023
AC-262,536 (category Selective androgen receptor modulators)
drug developed by Acadia Pharmaceuticals which acts as a selective androgen receptor modulator (SARM). Chemically it possesses endo-exo isomerism, with...
4 KB (308 words) - 21:05, 8 February 2024
GTx-027 (category Selective androgen receptor modulators)
GTx-027 is a selective androgen receptor modulator (SARM) which was under development for or of potential interest in the treatment of breast cancer and...
9 KB (718 words) - 04:15, 23 January 2025
MK-4541 (category Selective androgen receptor modulators)
MK-4541 is a dual selective androgen receptor modulator (SARM) and 5α-reductase inhibitor (5α-RI) which has been of interest for the potential treatment...
9 KB (702 words) - 15:55, 28 October 2024
pharmacodynamics, bicalutamide acts as a selective antagonist of the androgen receptor (AR), the biological target of androgens like testosterone and dihydrotestosterone...
186 KB (20,584 words) - 21:52, 29 May 2025
maintenance of male characteristics in vertebrates by binding to androgen receptors. This includes the embryological development of the primary male sex...
29 KB (3,166 words) - 21:29, 27 March 2025
company working on drugs in the selective estrogen receptor modulator (SERM) and selective androgen receptor modulator (SARM) classes. Its drugs in development...
7 KB (627 words) - 22:13, 22 November 2024
Clomifene (category Selective estrogen receptor modulators)
unknown cause or who are pregnant. Clomifene is in the selective estrogen receptor modulator (SERM) family of medication and is a nonsteroidal medication...
48 KB (4,759 words) - 20:23, 29 May 2025
JNJ-26146900 (category Selective androgen receptor modulators)
JNJ-26146900 is a selective androgen receptor modulator (SARM) which was developed by Johnson & Johnson for the potential treatment of prostate cancer...
8 KB (647 words) - 04:22, 14 January 2025
RU-59063 (category Selective androgen receptor modulators)
RU-59063 is a nonsteroidal androgen or selective androgen receptor modulator (SARM) which was first described in 1994 and was never marketed. It was originally...
7 KB (498 words) - 08:57, 8 June 2025