Seviteronel (developmental codes VT-464 and, formerly, INO-464) is an experimental cancer medication which is under development by Viamet Pharmaceuticals...
11 KB (882 words) - 12:00, 13 July 2024
permanently (rather than competitively) disables CYP17A1, once it binds to it. Seviteronel (VT-464) is a novel CYP17A1 inhibitor which is aimed to avoid co-administration...
25 KB (2,704 words) - 16:37, 12 February 2025
include the CYP17A1 inhibitors ketoconazole, abiraterone acetate, and seviteronel, the CYP11A1 (P450scc) inhibitor aminoglutethimide, and the 5α-reductase...
161 KB (15,261 words) - 19:58, 29 May 2025
antiandrogens that target testosterone synthesis (abiraterone acetate and seviteronel) or AR nuclear translocation (enzalutamide, apalutamide, and darolutamide)...
19 KB (2,124 words) - 22:42, 25 March 2025
Cimetidine Darolutamide Enzalutamide Flutamide Ketoconazole Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins...
3 KB (299 words) - 21:20, 29 May 2025
Cimetidine Darolutamide Enzalutamide Flutamide Ketoconazole Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins...
13 KB (1,661 words) - 08:23, 23 May 2025
Rezvilutamide Ro 2-7239 Ro 5-2537 RU-22930 RU-56187 RU-57073 RU-58642 RU-58841 Seviteronel Thalidomide Topilutamide (fluridil) Valproic acid Vinclozolin YM-580...
76 KB (7,617 words) - 21:07, 2 June 2025
with no antigonadotropic activity. Abiraterone acetate Ketoconazole Seviteronel Aminoglutethimide Alfatradiol Dutasteride Epristeride Finasteride Saw...
5 KB (254 words) - 18:23, 18 September 2023
Cimetidine Darolutamide Enzalutamide Flutamide Ketoconazole Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins...
27 KB (2,332 words) - 22:20, 29 May 2025
Cimetidine Darolutamide Enzalutamide Flutamide Ketoconazole Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins...
191 KB (18,328 words) - 22:14, 29 May 2025
Cimetidine Darolutamide Enzalutamide Flutamide Ketoconazole Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins...
25 KB (2,033 words) - 22:26, 29 May 2025
Rezvilutamide Ro 2-7239 Ro 5-2537 RU-22930 RU-56187 RU-57073 RU-58642 RU-58841 Seviteronel Thalidomide Topilutamide (fluridil) Valproic acid Vinclozolin YM-580...
18 KB (1,666 words) - 00:20, 24 May 2025
Cimetidine Darolutamide Enzalutamide Flutamide Ketoconazole Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins...
670 bytes (191 words) - 05:47, 13 February 2022
Cimetidine Darolutamide Enzalutamide Flutamide Ketoconazole Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins...
27 KB (3,041 words) - 20:28, 25 May 2025
Cimetidine Darolutamide Enzalutamide Flutamide Ketoconazole Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins...
49 KB (4,675 words) - 21:46, 29 May 2025
may also be followed by in-development drugs such as proxalutamide and seviteronel. Bicalutamide is the generic name of the drug in English and French and...
221 KB (21,804 words) - 20:07, 29 May 2025
Cimetidine Darolutamide Enzalutamide Flutamide Ketoconazole Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins...
29 KB (3,166 words) - 21:29, 27 March 2025
Rezvilutamide Ro 2-7239 Ro 5-2537 RU-22930 RU-56187 RU-57073 RU-58642 RU-58841 Seviteronel Thalidomide Topilutamide (fluridil) Valproic acid Vinclozolin YM-580...
84 KB (8,683 words) - 16:28, 3 June 2025
and the newer drugs abiraterone acetate, orteronel, galeterone, and seviteronel. CYP17A1 inhibitors, such as abiraterone acetate, are primarily used...
5 KB (418 words) - 21:48, 24 November 2024
steroidogenesis inhibitors: aminoglutethimide, ketoconazole, orteronel, seviteronel, others Miscellaneous: tanaproget (progestogen), finerenone (antimineralocorticoid)...
5 KB (381 words) - 22:24, 27 April 2025
Cimetidine Darolutamide Enzalutamide Flutamide Ketoconazole Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins...
12 KB (878 words) - 20:10, 29 May 2025
Rezvilutamide Ro 2-7239 Ro 5-2537 RU-22930 RU-56187 RU-57073 RU-58642 RU-58841 Seviteronel Thalidomide Topilutamide (fluridil) Valproic acid Vinclozolin YM-580...
6 KB (531 words) - 15:59, 8 November 2024
Cimetidine Darolutamide Enzalutamide Flutamide Ketoconazole Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins...
67 KB (6,840 words) - 20:36, 29 May 2025
Cimetidine Darolutamide Enzalutamide Flutamide Ketoconazole Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins...
62 KB (5,616 words) - 02:28, 2 June 2025
Cimetidine Darolutamide Enzalutamide Flutamide Ketoconazole Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins...
49 KB (4,091 words) - 17:57, 21 May 2025
Rezvilutamide Ro 2-7239 Ro 5-2537 RU-22930 RU-56187 RU-57073 RU-58642 RU-58841 Seviteronel Thalidomide Topilutamide (fluridil) Valproic acid Vinclozolin YM-580...
130 KB (13,325 words) - 21:19, 30 May 2025
Cimetidine Darolutamide Enzalutamide Flutamide Ketoconazole Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins...
34 KB (3,263 words) - 19:59, 20 May 2025
Cimetidine Darolutamide Enzalutamide Flutamide Ketoconazole Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins...
31 KB (3,434 words) - 14:06, 12 December 2024
Cimetidine Darolutamide Enzalutamide Flutamide Ketoconazole Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins...
36 KB (3,346 words) - 22:14, 29 May 2025
Cimetidine Darolutamide Enzalutamide Flutamide Ketoconazole Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins...
72 KB (7,424 words) - 04:12, 2 June 2025