The 5-HT2 receptors are a subfamily of 5-HT receptors that bind the endogenous neurotransmitter serotonin (5-hydroxytryptamine, 5-HT). The 5-HT2 subfamily...
2 KB (166 words) - 00:47, 13 May 2022
of the 5-HT2 receptor family that binds the neurotransmitter serotonin (5-hydroxytryptamine, 5-HT). Like all 5-HT2 receptors, the 5-HT2B receptor is Gq/G11-protein...
82 KB (7,913 words) - 17:32, 28 May 2025
The 5-HT2A receptor is a subtype of the 5-HT2 receptor that belongs to the serotonin receptor family and functions as a G protein-coupled receptor (GPCR)...
131 KB (13,680 words) - 11:36, 9 June 2025
5-HT2C receptor is a subtype of the 5-HT2 receptor that binds the endogenous neurotransmitter serotonin (5-hydroxytryptamine, 5-HT). Like all 5-HT2 receptors...
51 KB (6,133 words) - 17:35, 28 May 2025
actions, such as induction of dopamine and norepinephrine and serotonin 5-HT2 receptor agonism, which contributes to their effects as well. It is thought that...
70 KB (6,753 words) - 20:17, 18 June 2025
Chamomile (ethanol extract) 5-HT receptor 5-HT1 receptor 5-HT2 receptor 5-HT3 receptor 5-HT5 receptor 5-HT6 receptor 5-HT7 receptor GRCh38: Ensembl release...
18 KB (2,096 words) - 04:06, 20 May 2025
serotonin receptor agonist is an agonist of one or more serotonin receptors. They activate serotonin receptors in a manner similar to that of serotonin (5-hydroxytryptamine;...
16 KB (1,664 words) - 07:32, 20 February 2025
incontinence. The 5-HT2C receptors are one of three subtypes that belong to the serotonin 5-HT2 receptor subfamily along with 5-HT2A and 5-HT2B receptors. The development...
49 KB (5,040 words) - 23:14, 19 June 2025
of 5-HT3 receptors in cell lines and native tissues quickly followed. 5-HT1 receptor 5-HT2 receptor 5-HT4 receptor 5-HT5 receptor 5-HT6 receptor 5-HT7...
23 KB (2,440 words) - 22:20, 30 May 2025
Mirtazapine (category H1 receptor antagonists)
antidepressant drugs. Antagonism of the 5-HT2 subfamily of receptors and inverse agonism of the 5-HT2C receptor appears to be in part responsible for mirtazapine's...
90 KB (8,010 words) - 22:44, 8 June 2025
there is no 5-HT1C receptor since, after the receptor was cloned and further characterized, it was found to have more in common with the 5-HT2 family of...
65 KB (5,273 words) - 08:55, 28 May 2025
generalization of 5-MeO-DMT to the selective serotonin 5-HT2 receptor agonist (–)-DOM in animals. In accordance with the preceding findings, 5-MeO-DMT is reported...
72 KB (6,248 words) - 02:27, 22 June 2025
articles of the individual subtypes: 5-HT2 receptor 5-HT3 receptor 5-HT4 receptor 5-HT5 receptor 5-HT6 receptor 5-HT7 receptor Hoyer D, Clarke DE, Fozard JR...
5 KB (472 words) - 15:42, 23 May 2025
Paliperidone Risperidone 5-HT receptor 5-HT1 receptor 5-HT2 receptor 5-HT3 receptor 5-HT4 receptor 5-HT5 receptor 5-HT6 receptor GRCh38: Ensembl release...
26 KB (3,078 words) - 21:46, 20 May 2025
specifically at 5-HT2 receptor subtypes was proposed by Glennon et al. (1983c) based on drug discrimination studies in rats showing that the 5-HT2 antagonists...
94 KB (10,233 words) - 02:15, 29 June 2025
Ketanserin (category H1 receptor antagonists)
antiserotonergic agent in the study of the serotonin system; specifically, the 5-HT2 receptor family. The drug is taken by mouth. Side effects of ketanserin include...
30 KB (2,442 words) - 23:32, 17 June 2025
This is a list of miscellaneous agonists of the serotonin receptor subtype 5-HT2A (and other 5-HT2 subtypes to a varying extent) that fall outside the common...
30 KB (2,006 words) - 04:15, 14 June 2025
growth hormone, and β-endorphin. The receptor does not affect vasopressin or renin secretion, unlike the 5-HT2 receptors. It has been suggested that oxytocin...
59 KB (6,182 words) - 23:06, 22 May 2025
cocaine-conditioned rats, though 5-HT3's role is unclear. The 5-HT2 receptor (particularly the subtypes 5-HT2A, 5-HT2B and 5-HT2C) are involved in the locomotor-activating...
171 KB (17,561 words) - 13:32, 29 June 2025
5-methoxy analogue mebfap (5-MeO-3-APB; a benzofuran analogue of 5-MeO-AMT), which is known to have high affinity for the serotonin 5-HT2 receptors....
8 KB (719 words) - 20:06, 18 June 2025
Serotonin (redirect from 5-Hydroxytryptamine)
serotonin receptors, including the serotonin 5-HT1 (1A, 1B, 1D, 1E, 1F), 5-HT2 (2A, 2B, 2C), 5-HT3, 5-HT4, 5-HT5 (5A, 5B), 5-HT6, and 5-HT7 receptors. Except...
173 KB (18,295 words) - 19:45, 2 June 2025
Cyproheptadine (category 5-HT2 antagonists)
to ensure blockade of the 5-HT2 receptors for serotonin syndrome is 20 to 30 mg. Blockade of the serotonin 5-HT2B receptor may be specifically involved...
28 KB (2,279 words) - 15:24, 23 June 2025
7,N,N-TMT (category Serotonin receptor agonists)
derivative which acts as an agonist of 5-HT2 receptors. In animal tests, both 7-TMT and its 5-methoxy derivative 5-MeO-7-TMT produced behavioural responses...
4 KB (277 words) - 02:15, 11 April 2025
depression. αMS is a non-selective serotonin receptor agonist, including of the serotonin 5-HT2 receptors, and has been described as a "substitute neurotransmitter"...
10 KB (786 words) - 13:38, 11 April 2025
as a releaser of other monoamines and 5-HT2 receptor family agonist, similar to older compounds such as 5-APDB. 5-MAPDB was banned in the UK in June 2013...
4 KB (317 words) - 06:49, 8 May 2025
serotonin 5-HT1A receptor (Ki = 7.1 nM), the serotonin 5-HT1B receptor (Ki = 4,300 nM), and the serotonin 5-HT2 receptor (Ki = 1.0–450 nM). 5-HO-DPT was not...
4 KB (287 words) - 04:42, 19 June 2025
Locomotor activity (section Dopamine receptor agonists)
1007/BF01276460. PMID 8748668. O'Neill MF, Heron-Maxwell CL, Shaw G (June 1999). "5-HT2 receptor antagonism reduces hyperactivity induced by amphetamine, cocaine, and...
114 KB (12,382 words) - 04:41, 2 June 2025
5-HT1 or 5-HT2 receptors alone. Instead, a combination of actions at these and/or other receptors may be involved in its stimulus effects. α-Methyl-5-hydroxytryptophan...
24 KB (2,334 words) - 18:29, 20 May 2025
MDMA (redirect from (RS)-1-(1,3-Benzodioxol-5-yl)-N-methylpropan-2-amine)
other receptors. It is a low-potency partial agonist of the serotonin 5-HT2 receptors, including of the serotonin 5-HT2A, 5-HT2B, and 5-HT2C receptors. The...
250 KB (23,605 words) - 05:29, 28 June 2025
relation to Parkinson's disease. 5-HT receptor 5-HT1 receptor 5-HT2 receptor 5-HT3 receptor 5-HT4 receptor 5-HT5 receptor GRCh38: Ensembl release 89: ENSG00000158748...
29 KB (3,306 words) - 05:19, 25 May 2025