The adenosine A2A receptor, also known as ADORA2A, is an adenosine receptor, and also denotes the human gene encoding it. This protein is a member of...

four known types of adenosine receptors in humans: A1, A2A, A2B and A3; each is encoded by a different gene. The adenosine receptors are commonly known...

Adenosine A2A receptor antagonists are a class of drugs that block adenosine at the adenosine A2A receptor. Notable adenosine A2A receptor antagonists...

Cellular signaling by adenosine occurs through four known adenosine receptor subtypes (A1, A2A, A2B, and A3). Extracellular adenosine concentrations from...

subtypes of adenosine A2 receptors are known. Both are G protein-coupled adenosine receptors: Adenosine A2A receptor Adenosine A2B receptor This disambiguation...

D1–adenosine A1 D2–adenosine A2A D2–ghrelin receptor D2sh–TAAR1 (an autoreceptor heteromer) D4–adrenoceptor α1B D4–adrenoceptor β1 Dopamine receptor D1...

The adenosine A1 receptor (A1AR) is one member of the adenosine receptor group of G protein-coupled receptors with adenosine as endogenous ligand. A1 receptors...

enkephalin and a high density of dopamine D2 and adenosine A2A receptors (they also express adenosine A1 receptors), while dynorphinergic MSNs connect the striatum...

one adenosine A1 receptor and one dopamine D1 receptor) and the A2A–D2 receptor heterotetramer (this is a receptor complex with two adenosine A2A receptors...

A2A is an Italian company. A2A may also refer to: The Algonquin to Adirondacks Collaborative (A2A) The adenosine A2A receptor The UK Access to Archives...

ATL146e (A2A selective) PD81,723 (A1 allosteric enhancer) CF102 (Adenosine A3 receptor) Rosmarinic acid (A1 agonist) 5′-(N-Ethylcarboxamido)adenosine (NECA)...

the adenosine receptors (including A1, A2A, A2B, and A3). Conversely, agents like istradefylline and preladenant are selective adenosine A2A receptor antagonists...

(KW-6356) is a non-xanthine selective antagonist/inverse agonist of the adenosine A2A receptor that was previously under development by Kyowa Kirin as a monotherapy...

subset of these neurons that expresses both D2-type dopamine receptors and adenosine A2A receptors), located within the striatum the ventrolateral preoptic...

with antipsychotics for the management of schizophrenia. Giving an adenosine A2A receptor antagonist on top of existing treatment for Parkinson's disease...

Therapeutics for an undisclosed sum, as well as licensing PBF-509, an adenosine A2A receptor antagonist which is in Phase I clinical trials for non-small cell...

MSX-3 is a selective adenosine A2A receptor antagonist used in scientific research. Similarly to MSX-4, it is a water-soluble ester prodrug of MSX-2. MSX-3...

the DP1-dependent stimulation of adenosine formation and subsequent simulation of the adenosine A2A receptor by adenosine. In humans, a genetic variant of...

the adenosine A2A receptor, 410 nM for the adenosine A1 receptor (69-fold lower than for the A2A receptor), 260 nM for the adenosine A2B receptor (44-fold...

selective adenosine A2A receptor antagonist used in scientific research. It is a xanthine and a derivative of the non-selective adenosine receptor antagonist...

The adenosine A2B receptor, also known as ADORA2B, is a G-protein coupled adenosine receptor, and also denotes the human adenosine A2b receptor gene which...

(common cold). Istradefylline is a selective antagonist at the adenosine A2A receptor (A2AR), but the precise mechanism by which it exerts its therapeutic...

D2-type dopamine receptors, adenosine A2A receptors (A2A), DRD2–A2A heterotetramers, and enkephalin. Both types express glutamate receptors (NMDAR and AMPAR)...

5'-(N-Ethylcarboxamido)adenosine (NECA) is a nucleoside that is a non-selective adenosine receptor agonist. It has been used as a biochemical tool in...

Gao ZG, et al. (April 2011). "Structure of an agonist-bound human A2A adenosine receptor". Science. 332 (6027): 322–7. Bibcode:2011Sci...332..322X. doi:10...

Schering-Plough which acts as a potent and selective antagonist of the adenosine A2A receptor. It was being researched as a potential treatment for Parkinson's...

The adenosine A3 receptor, also known as ADORA3, is an adenosine receptor, but also denotes the human gene encoding it. Adenosine A3 receptors are G protein-coupled...

to an adenosine stress test, as it is a competitive antagonist of the A2A adenosine receptor and can attenuate the vasodilatory effects adenosine.[citation...

an experimental drug which acts as a selective inhibitor of the adenosine A2A receptor. It is in clinical trials for the treatment of lung cancer, and...

into P1 adenosine receptors and P2 nucleotide (ATP, ADP) receptors. P2 receptors were later subdivided into P2X, P2Y, P2T, and P2Z receptors. Subclasses...