The cannabinoid receptor 2 (CB2), is a G protein-coupled receptor from the cannabinoid receptor family that in humans is encoded by the CNR2 gene. It...
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Cannabinoid receptors, located throughout the body, are part of the endocannabinoid system of vertebrates– a class of cell membrane receptors in the G...
32 KB (3,086 words) - 18:05, 24 February 2025
membrane-bound receptors. The discovery of the first cannabinoid receptors in the 1980s helped to resolve this debate. These receptors are common in animals...
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A cannabinoid receptor antagonist, also known simply as a cannabinoid antagonist or as an anticannabinoid, is a type of cannabinoidergic drug that binds...
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Endocannabinoid system (redirect from Endogenous cannabinoid system)
endocannabinoids, which are neurotransmitters that bind to cannabinoid receptors, and cannabinoid receptor proteins that are expressed throughout the central...
68 KB (7,775 words) - 07:55, 31 May 2025
Cannabinoid receptor 1 (CB1), is a G protein-coupled cannabinoid receptor that in humans is encoded by the CNR1 gene. And discovered, by determination...
42 KB (4,352 words) - 07:40, 17 May 2025
has an entirely different chemical structure. WIN 55,212-2 is a potent cannabinoid receptor agonist that has been found to be a potent analgesic in a...
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Arachidonylcyclopropylamide (category Cannabinoids)
(ACPA) is a synthetic agonist of the cannabinoid receptor 1 (CB1R). ACPA is considered to be a selective cannabinoid agonist as it binds primarily to the...
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dose-dependent buildup of cannabinoids and related effects of cannabinoid toxicity the functionality of cannabinoid receptors in the brain and particularly...
38 KB (4,120 words) - 08:59, 25 May 2025
Synthetic cannabinoids, or neocannabinoids, are a class of designer drug molecules that bind to the same receptors to which cannabinoids (THC, CBD and...
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1999). "Evidence that the cannabinoid CB1 receptor is a 2-arachidonoylglycerol receptor. Structure-activity relationship of 2-arachidonoylglycerol, ether-linked...
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protein-coupled receptors (GPCRs), also known as seven-(pass)-transmembrane domain receptors, 7TM receptors, heptahelical receptors, serpentine receptors, and G...
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"Differential expression of cannabinoid receptors in the human colon: cannabinoids promote epithelial wound healing". Gastroenterology. 129 (2): 437–53. doi:10.1053/j...
103 KB (11,368 words) - 14:52, 2 June 2025
receptor (PTAFR, PAFR) InterPro: IPR002282 Cannabinoid receptor InterPro: IPR002230 Cannabinoid receptor 1 (brain) (CNR1, CB1R) Cannabinoid receptor 2...
25 KB (2,172 words) - 01:01, 29 November 2023
is the compound's binding affinity for the cannabinoid receptor type 1 (CB1) or cannabinoid receptor type 2 (CB2). Manera C, Tuccinardi T, Martinelli A...
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homebuilt aircraft CX5, identifier for Cannabinoid receptor type 2, a G protein-coupled receptor from the cannabinoid receptor family (6724) 1991 CX5, a main-belt...
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and a range of other health problems. While synthetic cannabinoids bind to the cannabinoid receptors in the body like natural cannabis, they are more aggressive...
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SR-144,528 (category Cannabinoid stubs)
selective antagonist of the CB2 cannabinoid receptor". The Journal of Pharmacology and Experimental Therapeutics. 284 (2): 644–50. PMID 9454810. Portier...
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Onternabez (category HU cannabinoids)
is a synthetic cannabinoid that acts as a potent cannabinoid agonist. It is highly selective for the cannabinoid-2 receptor (CB2 receptor) subtype, with...
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Cannabigerol (category Alpha-2 adrenergic receptor agonists)
of other cannabinoids, like THC and CBD. The pharmacodynamics of CBG are complex. It is a relatively weak ligand of the cannabinoid receptors, where it...
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tetrahydrocannabinol (THC) and tetrahydrocannabivarin (THCV), with total cannabinoid levels being much higher than observed in industrial hemp varieties....
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Are Influenced by Controlled Acute Administration". Cannabis and Cannabinoid Research. 2 (1): 217–223. doi:10.1089/can.2017.0024. PMC 5628568. PMID 29082319...
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frequency than the norm. Cannabinoids produce a "marked depression of motor activity" via activation of neuronal cannabinoid receptors belonging to the CB1...
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AM-2201 (redirect from AM4 (cannabinoid))
potent but nonselective full agonist for the cannabinoid receptor. It is part of the AM series of cannabinoids discovered by Alexandros Makriyannis at Northeastern...
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AM-694 (category AM cannabinoids)
(1-(5-fluoropentyl)-3-(2-iodobenzoyl)indole) is a designer drug that acts as a potent and selective agonist for the cannabinoid receptor CB1. It is used in...
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AM-1241 (category AM cannabinoids)
selective agonist for the cannabinoid receptor CB2, with a Ki of 3.4 nM at CB2 and 80 times selectivity over the related CB1 receptor. It has analgesic effects...
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389–462. doi:10.1124/pr.58.3.2. PMC 2241751. PMID 16968947. Hongfeng Deng. Design and synthesis of selective cannabinoid receptor ligands: Aminoalkylindole...
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ADB-BUTINACA (category Cannabinoids)
acid-derived synthetic cannabinoid receptor agonists related to ADB-BUTINACA, APP-BUTINACA, and ADB-P7AICA". RSC Medicinal Chemistry. 13 (2): 156–174. doi:10...
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212-2 Pharmacology Cannabinoid receptors Cannabinoid receptor type 1 Cannabinoid receptor type 2 Endocannabinoids (activate cannabinoid receptors) 2-AG...
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Synthetic drug (section Synthetic cannabinoids)
To exert the psychoactive effect, specific receptors such as cannabinoid, dopamine and serotonin receptors are either stimulated or inhibited There are...
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