• Thumbnail for Peroxisome proliferator-activated receptor
    field of molecular biology, the peroxisome proliferatoractivated receptors (PPARs) are a group of nuclear receptor proteins that function as transcription...
    18 KB (1,885 words) - 06:27, 15 April 2025
  • Thumbnail for Peroxisome proliferator-activated receptor gamma
    Peroxisome proliferator-activated receptor gamma (PPAR-γ or PPARG), also known as the glitazone reverse insulin resistance receptor, or NR1C3 (nuclear...
    19 KB (2,091 words) - 05:22, 13 July 2024
  • Thumbnail for Peroxisome proliferator-activated receptor alpha
    proliferator-activated receptor delta and peroxisome proliferator-activated receptor gamma, PPAR-alpha is part of the subfamily of peroxisome proliferator-activated receptors...
    22 KB (2,602 words) - 18:54, 1 May 2025
  • Thumbnail for Peroxisome proliferator-activated receptor delta
    Peroxisome proliferator-activated receptor delta (PPAR-delta), or (PPAR-beta), also known as Nuclear hormone receptor 1 (NUC1) is a nuclear receptor that...
    18 KB (1,963 words) - 10:40, 5 February 2025
  • proposed to be the peroxisome proliferator-activated receptor alpha (PPAR-α). PEA also has affinity to cannabinoid-like G-coupled receptors GPR55 and GPR119...
    47 KB (5,040 words) - 12:26, 11 January 2025
  • Thumbnail for PPAR agonist
    PPAR agonists are drugs which act upon the peroxisome proliferator-activated receptor. They are used for the treatment of symptoms of the metabolic syndrome...
    10 KB (1,219 words) - 10:05, 30 March 2025
  • Thumbnail for Telmisartan
    Telmisartan (category Angiotensin II receptor antagonists)
    from PPAR-γ. Telmisartan's activity at the peroxisome proliferator-activated receptor delta (PPAR-δ) receptor has prompted speculation around its potential...
    19 KB (1,699 words) - 20:43, 1 April 2025
  • Thumbnail for Pparg coactivator 1 alpha
    Peroxisome proliferator-activated receptor gamma coactivator 1-alpha (PGC-1α) is a protein that in humans is encoded by the PPARGC1A gene. PPARGC1A is...
    32 KB (3,869 words) - 14:22, 16 January 2025
  • Thumbnail for GW501516
    expression of GLUT1 and SLC1A5. Acadesine GFT505 GW0742 Irisin Peroxisome proliferator-activated receptor Sodelglitazar SR9009 Koh B (2013-03-22). "Anti-doping...
    21 KB (2,027 words) - 03:42, 10 May 2025
  • Thumbnail for Estrogen-related receptor alpha
    Kelly DP (October 2004). "Estrogen-related receptor alpha directs peroxisome proliferator-activated receptor alpha signaling in the transcriptional control...
    17 KB (1,995 words) - 19:11, 3 February 2025
  • Another potential target of antiepileptic drugs is the peroxisome proliferator-activated receptor alpha. Some anticonvulsants have shown antiepileptogenic...
    71 KB (5,805 words) - 11:51, 5 May 2025
  • Thumbnail for Seladelpar
    used as the lysine dihydrate salt. It is a peroxisome proliferator-activated receptor delta (PPARδ) receptor agonist. The compound was licensed from Janssen...
    9 KB (547 words) - 03:47, 4 March 2025
  • Thumbnail for Farnesoid X receptor
    Farnesoid X receptor has been shown to interact with: Peroxisome proliferator-activated receptor gamma coactivator 1-alpha and Retinoid X receptor alpha. A number...
    18 KB (2,072 words) - 23:27, 23 April 2025
  • Thumbnail for Elafibranor
    active metabolite GFT1007 are peroxisome proliferator-activated receptor (PPAR) agonists, both of which activate PPAR-alpha, PPAR-gamma, and PPAR-delta...
    15 KB (984 words) - 20:57, 9 May 2025
  • Thumbnail for Fibrate
    increased risk of rhabdomyolysis. Fibrates stimulate peroxisome proliferator activated receptor (PPAR) alpha, which controls the expression of gene products...
    10 KB (1,091 words) - 01:14, 8 October 2024
  • Thumbnail for Thiazolidinedione
    Thiazolidinediones or TZDs act by activating PPARs (peroxisome proliferator-activated receptors), a group of nuclear receptors, specific for PPARγ (PPAR-gamma...
    20 KB (2,167 words) - 15:36, 9 January 2025
  • Thumbnail for Ciglitazone
    (February 1996). "The structure-activity relationship between peroxisome proliferator-activated receptor gamma agonism and the antihyperglycemic activity of thiazolidinediones"...
    6 KB (424 words) - 09:21, 4 August 2023
  • Thumbnail for Pirinixic acid
    Pirinixic acid is a peroxisome proliferator-activated receptor alpha (PPARα) agonist that is under experimental investigation for prevention of severe...
    7 KB (675 words) - 00:08, 26 March 2025
  • Thumbnail for Gemfibrozil
    lipolysis. It does so by activating peroxisome proliferator-activated receptor alpha (PPARα) 'transcription factor ligand', a receptor that is involved in...
    12 KB (927 words) - 02:17, 2 December 2024
  • Thumbnail for Ibuprofen
    cord injury. Another unusual activity is inhibition of the sweet taste receptor. After oral administration, peak serum concentration is reached after 1–2 hours...
    67 KB (6,231 words) - 12:45, 16 May 2025
  • Thumbnail for Genistein
    Genistein (category Glycine receptor antagonists)
    the G protein-coupled estrogen receptor, and binds to and activates all three peroxisome proliferator-activated receptor isoforms, α, δ, and γ. Genistein...
    16 KB (1,473 words) - 06:11, 9 May 2025
  • Thumbnail for GW0742
    Roberts-Thomson SJ (July 2004). "Effect of the peroxisome proliferator-activated receptor beta activator GW0742 in rat cultured cerebellar granule neurons"...
    9 KB (827 words) - 19:19, 6 May 2024
  • Thumbnail for Liver X receptor alpha
    nuclear hormone receptor LXR alpha interacts with the peroxisome proliferator-activated receptor and inhibits peroxisome proliferator signaling". The...
    14 KB (1,645 words) - 21:40, 5 May 2025
  • Thumbnail for Saroglitazar
    a dual PPAR agonist at the subtypes α (alpha) and γ (gamma) of the peroxisome proliferator-activated receptor (PPAR). Agonist action on PPARα lowers high...
    9 KB (767 words) - 21:52, 3 March 2025
  • Thumbnail for Cholesterol 7 alpha-hydroxylase
    cultured cells is mediated via the liver x receptor alpha and peroxisome proliferator-activated receptor alpha heterodimer". Nucleic Acids Research. 32...
    22 KB (2,660 words) - 01:58, 10 March 2025
  • which act upon the peroxisome proliferator-activated receptor alpha This disambiguation page lists articles associated with the title Alpha agonist. If an...
    246 bytes (60 words) - 06:54, 14 August 2020
  • Thumbnail for Fatty liver disease
    "Molecular mechanisms of alcoholic fatty liver: role of peroxisome proliferator-activated receptor alpha". Alcohol. 34 (1): 35–8. doi:10.1016/j.alcohol.2004...
    38 KB (3,799 words) - 16:43, 10 May 2025
  • Thumbnail for Oleoylethanolamide
    Oleoylethanolamide (OEA) is an endogenous peroxisome proliferator-activated receptor alpha (PPAR-α) agonist. It is a naturally occurring ethanolamide lipid...
    9 KB (835 words) - 03:29, 7 April 2025
  • Thumbnail for Nuclear receptor coactivator 1
    PCAF, PPARGC1A, Peroxisome proliferator-activated receptor alpha, SNW1, STAT3, STAT6, TRIP4, and Thyroid hormone receptor beta. GRCh38: Ensembl release...
    14 KB (1,625 words) - 14:43, 28 October 2024
  • Thumbnail for Retinoic acid receptor alpha
    (May 1999). "Identification of nuclear receptor corepressor as a peroxisome proliferator-activated receptor alpha interacting protein". The Journal of Biological...
    25 KB (2,847 words) - 00:27, 11 August 2024