The adenosine A2B receptor, also known as ADORA2B, is a G-protein coupled adenosine receptor, and also denotes the human adenosine A2b receptor gene which...

four known types of adenosine receptors in humans: A1, A2A, A2B and A3; each is encoded by a different gene. The adenosine receptors are commonly known...

subtypes of adenosine A2 receptors are known. Both are G protein-coupled adenosine receptors: Adenosine A2A receptor Adenosine A2B receptor This disambiguation...

Cellular signaling by adenosine occurs through four known adenosine receptor subtypes (A1, A2A, A2B, and A3). Extracellular adenosine concentrations from...

A2B may refer to: A2B, Adenosine A2B receptor A2B Australia, a taxi operator A2B Bicycles, an electric bicycle company A2B-online, an intermodal trailer...

The adenosine A2A receptor, also known as ADORA2A, is an adenosine receptor, and also denotes the human gene encoding it. This protein is a member of...

Biginelli reaction have been investigated as potential selective Adenosine A2b receptor antagonists. Including highly selective tricyclic compounds. The...

The adenosine A1 receptor (A1AR) is one member of the adenosine receptor group of G protein-coupled receptors with adenosine as endogenous ligand. A1 receptors...

An adenosine receptor antagonist is a drug which acts as an antagonist of one or more of the adenosine receptors. The best known are xanthines and their...

four adenosine receptor subtypes (A1, A2A, A2B, and A3), although with varying potencies. The affinity (KD) values of caffeine for the human adenosine receptors...

The adenosine A3 receptor, also known as ADORA3, is an adenosine receptor, but also denotes the human gene encoding it. Adenosine A3 receptors are G protein-coupled...

into P1 adenosine receptors and P2 nucleotide (ATP, ADP) receptors. P2 receptors were later subdivided into P2X, P2Y, P2T, and P2Z receptors. Subclasses...

the adenosine A2A receptor, 410 nM for the adenosine A1 receptor (69-fold lower than for the A2A receptor), 260 nM for the adenosine A2B receptor (44-fold...

the adenosine receptors (including A1, A2A, A2B, and A3). Conversely, agents like istradefylline and preladenant are selective adenosine A2A receptor antagonists...

D1–adenosine A1 D2–adenosine A2A D2–ghrelin receptor D2sh–TAAR1 (an autoreceptor heteromer) D4–adrenoceptor α1B D4–adrenoceptor β1 Dopamine receptor D1...

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline)...

Tobias (June 2013). "Attenuating myocardial ischemia by targeting A2B adenosine receptors". Trends in Molecular Medicine. 19 (6): 345–354. doi:10.1016/j...

protein-coupled receptors (GPCRs), also known as seven-(pass)-transmembrane domain receptors, 7TM receptors, heptahelical receptors, serpentine receptors, and G...

lower affinity to A2A and A2B receptors causing dilation of efferent arterioles. The binding of adenosine to the A1 receptor causes a complex signal cascade...

Cell surface receptors (membrane receptors, transmembrane receptors) are receptors that are embedded in the plasma membrane of cells. They act in cell...

Muscarinic acetylcholine receptors (mAChRs) are acetylcholine receptors that form G protein-coupled receptor complexes in the cell membranes of certain...

adenosine, which triggers intracellular signal transduction via both adenosine A1 receptors and two sub-types of adenosine A2 receptors (A2A and A2B receptors)...

"Inhibition of tPA-induced hemorrhagic transformation involves adenosine A2b receptor activation after cerebral ischemia". Neurobiol Dis. 108: 173–182...

a selective non-xanthinic adenosine A2B receptor antagonist. Discovered in 2016, it has a Ki of 3.49 nM on the A2B receptor and >1000-fold selectivity...

lung tissue. Some benzodiazepines have inhibitory effects on the adenosine A2B receptor mediated secretion of IL-8 in human mast cells. In a 2013 study...

antagonist at adenosine receptors. d9-Caffeine was assessed for human adenosine receptor antagonism at the four receptor subtypes: A1, A2A, A2B, and A3, and...

PMID 23601906. Sepúlveda C, Palomo I, Fuentes E (2016). "Role of adenosine A2b receptor overexpression in tumor progression". Life Sciences. 166: 92–99...

receptors on the neutrophil, and the affinity of these receptors for adenosine. Micromolar concentrations of adenosine activate A2A and A2B receptors...

The μ-opioid receptors (MOR) are a class of opioid receptors with a high affinity for enkephalins and beta-endorphin, but a low affinity for dynorphins...

four well-known adenosine receptors found in the body, A1, A2A, A2B, and A3. The endogenous agonist for these receptors is adenosine, which is a purine...