Testolactone (INNTooltip International Nonproprietary Name, USANTooltip United States Adopted Name) (brand name Teslac) is a non-selective, irreversible...
10 KB (871 words) - 17:49, 11 November 2023
aminoglutethimide, arimistane, exemestane, formestane, letrozole, and testolactone Selective estrogen receptor modulators (SERMs), including bazedoxifene...
9 KB (701 words) - 20:01, 1 January 2025
Examples of substances under this schedule: All insulin preparations, testolactone, hydroxyurea, daunorubicin, metformin, diphenhydramine, carbutamide,...
11 KB (1,007 words) - 10:06, 19 February 2025
inhibitors (AIs) include: Aminoglutethimide (Elipten, Cytadren, Orimeten) Testolactone (Teslac) Anastrozole (Arimidex) Letrozole (Femara) Exemestane (Aromasin)...
21 KB (2,089 words) - 16:27, 23 May 2025
steroidogenesis, such as cyproterone acetate, ketoconazole, spironolactone, and testolactone. Alternatively, the combination of the androgen receptor antagonist bicalutamide...
4 KB (323 words) - 03:08, 16 October 2024
anastrozole, letrozole, aminoglutethimide, exemestane, formestane, and testolactone are banned. Selective estrogen receptor modulators, including raloxifene...
20 KB (1,822 words) - 20:19, 13 December 2024
indication for use of aromatase inhibitors improving spermatogenesis, testolactone has been shown to be effective when compared to placebo. Though there...
23 KB (2,599 words) - 01:55, 14 April 2024
antagonists ERA (Atrasentan) Retinoid X receptor (Bexarotene) Sex steroid (Testolactone) Other/ungrouped Adagrasib Aflibercept Arsenic trioxide Asparagine depleters...
34 KB (3,131 words) - 01:44, 25 May 2025
while Brunk was in possession of drug paraphernalia and nine tablets of testolactone. Both Szatkowski and Brunk were released after posting bail, and were...
175 KB (18,316 words) - 08:49, 19 May 2025
Fluoxymesterone (Halotestin) (1958) Dromostanolone (Drolban) (1961) Testolactone (Teslac) (1970) Methyl prednisolone Prednisolone Zoladex (1989) Biologicals...
36 KB (3,029 words) - 05:59, 28 May 2025
antagonists ERA (Atrasentan) Retinoid X receptor (Bexarotene) Sex steroid (Testolactone) Other/ungrouped Adagrasib Aflibercept Arsenic trioxide Asparagine depleters...
30 KB (2,799 words) - 01:53, 30 May 2025
antagonists ERA (Atrasentan) Retinoid X receptor (Bexarotene) Sex steroid (Testolactone) Other/ungrouped Adagrasib Aflibercept Arsenic trioxide Asparagine depleters...
5 KB (324 words) - 08:56, 9 December 2024
inhibitors Generation Medication Dosage % inhibitiona Classb IC50c First Testolactone 250 mg 4x/day p.o. ? Type I ? 100 mg 3x/week i.m. ? Rogletimide 200 mg...
28 KB (2,356 words) - 19:57, 29 May 2025
Trilostane Aromatase inhibitors First-generation: Aminoglutethimide Testolactone Second-generation: Fadrozole Formestane Third-generation: Anastrozole...
73 KB (7,804 words) - 06:01, 13 May 2025
antagonists ERA (Atrasentan) Retinoid X receptor (Bexarotene) Sex steroid (Testolactone) Other/ungrouped Adagrasib Aflibercept Arsenic trioxide Asparagine depleters...
24 KB (2,272 words) - 20:10, 29 May 2025
antagonists ERA (Atrasentan) Retinoid X receptor (Bexarotene) Sex steroid (Testolactone) Other/ungrouped Adagrasib Aflibercept Arsenic trioxide Asparagine depleters...
20 KB (1,615 words) - 21:06, 24 April 2025
antagonists ERA (Atrasentan) Retinoid X receptor (Bexarotene) Sex steroid (Testolactone) Other/ungrouped Adagrasib Aflibercept Arsenic trioxide Asparagine depleters...
27 KB (2,446 words) - 16:23, 8 May 2025
antagonists ERA (Atrasentan) Retinoid X receptor (Bexarotene) Sex steroid (Testolactone) Other/ungrouped Adagrasib Aflibercept Arsenic trioxide Asparagine depleters...
40 KB (3,616 words) - 12:21, 23 May 2025
and led to the development of other aromatase inhibitors. Along with testolactone, it is described as a "first-generation" aromatase inhibitor. AG has...
32 KB (2,828 words) - 02:53, 12 January 2025
antagonists ERA (Atrasentan) Retinoid X receptor (Bexarotene) Sex steroid (Testolactone) Other/ungrouped Adagrasib Aflibercept Arsenic trioxide Asparagine depleters...
33 KB (3,152 words) - 18:41, 25 April 2025
antagonists ERA (Atrasentan) Retinoid X receptor (Bexarotene) Sex steroid (Testolactone) Other/ungrouped Adagrasib Aflibercept Arsenic trioxide Asparagine depleters...
5 KB (290 words) - 20:59, 6 January 2024
antagonists ERA (Atrasentan) Retinoid X receptor (Bexarotene) Sex steroid (Testolactone) Other/ungrouped Adagrasib Aflibercept Arsenic trioxide Asparagine depleters...
25 KB (2,517 words) - 19:48, 6 March 2025
antagonists ERA (Atrasentan) Retinoid X receptor (Bexarotene) Sex steroid (Testolactone) Other/ungrouped Adagrasib Aflibercept Arsenic trioxide Asparagine depleters...
45 KB (4,630 words) - 20:02, 29 May 2025
antagonists ERA (Atrasentan) Retinoid X receptor (Bexarotene) Sex steroid (Testolactone) Other/ungrouped Adagrasib Aflibercept Arsenic trioxide Asparagine depleters...
19 KB (1,730 words) - 06:30, 25 May 2025
antagonists ERA (Atrasentan) Retinoid X receptor (Bexarotene) Sex steroid (Testolactone) Other/ungrouped Adagrasib Aflibercept Arsenic trioxide Asparagine depleters...
11 KB (1,239 words) - 22:33, 24 May 2025
inhibitors Generation Medication Dosage % inhibitiona Classb IC50c First Testolactone 250 mg 4x/day p.o. ? Type I ? 100 mg 3x/week i.m. ? Rogletimide 200 mg...
22 KB (1,991 words) - 18:51, 24 May 2025
Teslac Teslac (Bristol-Myers Squibb) Teslascan Tessalon Testim Testoderm testolactone (INN) Testomar Testopel testosterone ketolaurate (INN) testosterone undecanoate...
14 KB (670 words) - 23:06, 2 May 2025
Trilostane Aromatase inhibitors First-generation: Aminoglutethimide Testolactone Second-generation: Fadrozole Formestane Third-generation: Anastrozole...
52 KB (4,098 words) - 13:29, 29 May 2025
antagonists ERA (Atrasentan) Retinoid X receptor (Bexarotene) Sex steroid (Testolactone) Other/ungrouped Adagrasib Aflibercept Arsenic trioxide Asparagine depleters...
12 KB (1,038 words) - 11:18, 27 May 2025
clomiphene citrate (an antiestrogen) and aromatase inhibitors such as testolactone or anastrozole have shown effectiveness in benefiting spermatogenesis...
63 KB (7,688 words) - 19:20, 23 May 2025