5-Hydroxytryptamine receptor 2B (5-HT2B) also known as serotonin receptor 2B is a protein that in humans is encoded by the HTR2B gene. 5-HT2B is a member...

5-HT2A receptor 5-HT2B receptor 5-HT2C receptor 5-HT1 receptor 5-HT3 receptor 5-HT4 receptor 5-HT5 receptor 5-HT6 receptor 5-HT7 receptor Category:5-HT2...

the 5-HT2A receptor like cyproheptadine and chlorpromazine are able to reverse and mediate recovery from serotonin syndrome. Agonists of the 5-HT2B receptor...

5-HT receptors, 5-hydroxytryptamine receptors, or serotonin receptors, are a group of G protein-coupled receptor and ligand-gated ion channels found in...

entities: the 5-HT2A (formerly known as 5-HT2 or D), the 5-HT2B (formerly known as 5-HT2F) and the 5-HT2C (formerly known as 5-HT1C) receptors. The 5-HT2A receptors...

to be potent serotonin 5-HT2B receptor agonists and others finding them to be very weak or negligible serotonin 5-HT2B receptor agonists, depending on...

the same type of serotonin receptor binding as pergolide. Although lisuride, a related drug, also binds to the 5-HT2B receptor, it acts as an antagonist...

Activation of the 5-HT2B receptor is a well-known antitarget and is associated with cardiac valvulopathy. However, not all 5-HT2B receptor agonists, for instance...

reuptake inhibitor (SNDRI). 5-APB is a potent agonist of the serotonin 5-HT2A and 5-HT2B receptors. Its EC50Tooltip half-maximal effective...

incontinence. The 5-HT2C receptors are one of three subtypes that belong to the serotonin 5-HT2 receptor subfamily along with 5-HT2A and 5-HT2B receptors. The development...

for the 5-HT1, GABA, mAChRs, α1-, and β-adrenoreceptors. It is a potent agonist of the 5-HT2B receptor, but shows biased agonism at this receptor and does...

Serotonin 5-HT2B receptor antagonists by themselves do not appear to affect locomotor activity. However, antagonists of the serotonin 5-HT2B receptor decrease...

In any case, in other research, serotonin 5-HT2B receptor knockout or selective serotonin 5-HT2B receptor antagonism with RS-127445 has been found to...

α2-adrenergic receptor antagonist. It has also been shown to function as a 5-HT1A receptor partial agonist and 5-HT2A and 5-HT2B receptor antagonist. Ajmalicine...

serotonin 5-HT2B receptor than the reference serotonin 5-HT2B receptor agonist, BW-723C86, which is commonly used for research into the serotonin 5-HT2B receptor...

Metatone) – also a 5-HT2A receptor antagonist Viloxazine (Qelbree, formerly Vivalan) – also a 5-HT2B receptor antagonist and 5-HT2C receptor agonist Atomoxetine...

acts as a potent and well-balanced serotonin 5-HT2A and 5-HT2C receptor agonist, serotonin 5-HT2B receptor antagonist, and serotonin releasing agent. It...

different receptors. Through 5-HT1B receptors, it negatively regulates bone mass, while it does so positively through 5-HT2B receptors and 5-HT2C receptors. There...

5-HT2A receptor (EC50Tooltip half-maximal effective concentration = 162 nM; EmaxTooltip maximal efficacy = 89%) and of the serotonin 5-HT2B receptor (EC50...

400-fold selective for the serotonin 5-HT2B receptor over the serotonin 5-HT2A and 5-HT2C receptors, respectively. 5-MT, in contrast to the closely related...

as a 5-HT2B receptor agonist. It has anxiolytic effects in animal studies, and is also used for investigating the function of the 5-HT2B receptor in a...

identified as 5-MeO-AMT. 5-MeO-AMT acts as a non-selective serotonin receptor agonist, including of the serotonin 5-HT1A, 5-HT2A, and 5-HT2B receptors, among...

5-HT2C receptor, with negligible affinity for the serotonin 5-HT2A and 5-HT2B receptors. Because it does not activate the serotonin 5-HT2B receptor,...

best-known and most significant antitargets are the hERG channel and the 5-HT2B receptor, both of which cause long-term problems with heart function that can...

Affecting 5-HT2B Receptors". 5-HT2B Receptors. The Receptors. Vol. 35. Cham: Springer International Publishing. pp. 277–289. doi:10.1007/978-3-030-55920-5_16...

the serotonin 5-HT2A receptor, it is also an antagonist of the serotonin 5-HT2B receptor and an agonist of the serotonin 5-HT2C receptor. The drug's route...

335 nM for the serotonin 5-HT2A receptor, 8.39 nM for the serotonin 5-HT2B receptor, and 82–84 nM for the serotonin 5-HT2C receptor. Its activational potencies...

serotonin 5-HT2 receptors have been found to be 0.40 nM for the serotonin 5-HT2A receptor, 24.5 to 35.0 nM for the serotonin 5-HT2B receptor, and 1.0 nM...

into the BLA significantly increased sociability. The serotonin 5-HT2B and 5-HT2C receptor antagonist SB-206553 has also been found to block MDMA-induced...

instead as 5-HT2B receptor agonists such as cabergoline and pergolide but is similar to lisuride which likewise acts as a 5-HT2B receptor antagonist....