• The 5-HT3 receptor belongs to the Cys-loop superfamily of ligand-gated ion channels (LGICs) and therefore differs structurally and functionally from all...
    22 KB (2,395 words) - 18:29, 18 July 2024
  • Thumbnail for 5-HT3 antagonist
    The 5-HT3 antagonists, informally known as "setrons", are a class of drugs that act as receptor antagonists at the 5-HT3 receptor, a subtype of serotonin...
    43 KB (4,628 words) - 09:00, 16 April 2025
  • Thumbnail for Serotonin receptor agonist
    individuals. 2-Methyl-5-hydroxytryptamine (2-methylserotonin) and quipazine are moderately selective agonists of the 5-HT3 receptor that are used in scientific...
    16 KB (1,664 words) - 07:32, 20 February 2025
  • 5-HT2A receptor 5-HT2B receptor 5-HT2C receptor 5-HT1 receptor 5-HT3 receptor 5-HT4 receptor 5-HT5 receptor 5-HT6 receptor 5-HT7 receptor Category:5-HT2...
    2 KB (166 words) - 00:47, 13 May 2022
  • Thumbnail for HTR3E
    HTR3E (category Transmembrane receptor stubs)
    5-hydroxytryptamine receptor 3E is a protein that in humans is encoded by the HTR3E gene. The protein encoded by this gene is a subunit of the 5-HT3 receptor...
    3 KB (324 words) - 22:12, 3 March 2023
  • Thumbnail for 5-HT receptor
    response. The exception to this is the 5-HT3 receptor which is a ligand-gated ion channel. In 2014, a novel 5-HT receptor was isolated from the small white butterfly...
    65 KB (5,270 words) - 07:14, 24 November 2024
  • Thumbnail for Ondansetron
    Ondansetron (category 5-HT3 antagonists)
    It is a serotonin 5-HT3 receptor antagonist. It does not have any effect on dopamine receptors or muscarinic acetylcholine receptor and therefore does...
    35 KB (3,291 words) - 06:02, 20 April 2025
  • Thumbnail for 5-HT7 receptor
    Paliperidone Risperidone 5-HT receptor 5-HT1 receptor 5-HT2 receptor 5-HT3 receptor 5-HT4 receptor 5-HT5 receptor 5-HT6 receptor GRCh38: Ensembl release...
    25 KB (2,993 words) - 19:47, 5 January 2025
  • D2 receptors, serotonin 5-HT3 receptors, opioid receptors, acetylcholine receptors, and receptors for substance P. Stimulation of different receptors are...
    22 KB (2,403 words) - 02:48, 4 September 2023
  • subclass consists of drugs selectively acting at the 5-HT3 receptors, and thus are known as 5-HT3 antagonists. They are efficacious in treating chemotherapy-induced...
    5 KB (503 words) - 05:28, 26 March 2025
  • Thumbnail for Monoamine receptor
    monoamine structure. The monoamine receptors are almost all G protein-coupled receptors, with the serotonin 5-HT3 receptor being a notable exception as a...
    2 KB (163 words) - 11:14, 6 November 2023
  • Thumbnail for 5-HT6 receptor
    relation to Parkinson's disease. 5-HT receptor 5-HT1 receptor 5-HT2 receptor 5-HT3 receptor 5-HT4 receptor 5-HT5 receptor GRCh38: Ensembl release 89: ENSG00000158748...
    29 KB (3,306 words) - 04:01, 15 May 2025
  • Thumbnail for 5-HT2A receptor
    label two different 5-HT receptors, and neither of them displaced morphine, leading to naming of the 5-HT1, 5-HT2 and 5-HT3 receptors, corresponding to...
    128 KB (13,443 words) - 21:15, 18 May 2025
  • Thumbnail for Mirtazapine
    Mirtazapine (category H1 receptor antagonists)
    antagonism of the serotonin 5-HT2A and 5-HT2C receptors, while the (R)-(–) enantiomer is responsible for antagonism of the 5-HT3 receptor. Both enantiomers are...
    90 KB (8,058 words) - 23:40, 12 May 2025
  • sickness and the more serious hyperemesis gravidarum. 5-HT3 receptor antagonists block serotonin receptors in the central nervous system and gastrointestinal...
    16 KB (1,746 words) - 04:11, 6 February 2025
  • Thumbnail for 5-HT4 receptor
    Chamomile (ethanol extract) 5-HT receptor 5-HT1 receptor 5-HT2 receptor 5-HT3 receptor 5-HT5 receptor 5-HT6 receptor 5-HT7 receptor GRCh38: Ensembl release...
    18 KB (2,075 words) - 06:39, 29 April 2025
  • dopamine, histamine (H1 receptor), substance P (NK-1 receptor), and serotonin (5-HT3 receptor). There are also opioid receptors present, which may be involved...
    17 KB (2,454 words) - 13:11, 18 April 2025
  • Thumbnail for HTR3D
    HTR3D (category Transmembrane receptor stubs)
    5-hydroxytryptamine receptor 3D is a protein that in humans is encoded by the HTR3D gene. The protein encoded by this gene is a subunit of the 5-HT3 receptor...
    2 KB (196 words) - 22:12, 3 March 2023
  • Thumbnail for HTR3A
    HTR3A (category Transmembrane receptor stubs)
    transcript variants encoding different isoforms have been identified. 5-HT3 receptor GRCh38: Ensembl release 89: ENSG00000166736 – Ensembl, May 2017 GRCm38:...
    8 KB (996 words) - 08:26, 29 April 2025
  • Thumbnail for 5-HT5A receptor
    206 nM affinity. SB-699,551 5-HT receptor 5-HT1 receptor 5-HT2 receptor 5-HT3 receptor 5-HT4 receptor 5-HT6 receptor 5-HT7 receptor GRCh38: Ensembl release...
    16 KB (1,773 words) - 06:08, 29 April 2025
  • Thumbnail for HTR3C
    HTR3C (category Transmembrane receptor stubs)
    5-hydroxytryptamine receptor 3C is a protein that in humans is encoded by the HTR3C gene. The protein encoded by this gene is a subunit of the 5-HT3 receptor...
    2 KB (276 words) - 22:12, 3 March 2023
  • Thumbnail for 2-Methyl-5-hydroxytryptamine
    moderately selective full agonist at the 5-HT3 receptor. 5-Carboxamidotryptamine 5-Methoxytryptamine α-Methyl-5-hydroxytryptamine Elz S, Zimmermann H, Rehse...
    3 KB (188 words) - 07:27, 27 March 2025
  • loss, or improving absorption. There are four main classes: opiates, 5-HT3 receptor antagonists, adsorbents, and bulk-forming agents. Commonly used medications...
    10 KB (854 words) - 20:58, 6 May 2025
  • Thumbnail for Bufotenin
    Bufotenin (redirect from 5-OH-DMT)
    potent and non-selective serotonin receptor agonist, including of the serotonin 5-HT1A, 5-HT2A, 5-HT2C, and 5-HT3 receptors, among others. It also acts as...
    91 KB (8,913 words) - 00:23, 18 May 2025
  • Thumbnail for Serotonin
    serotonin receptors, including the serotonin 5-HT1 (1A, 1B, 1D, 1E, 1F), 5-HT2 (2A, 2B, 2C), 5-HT3, 5-HT4, 5-HT5 (5A, 5B), 5-HT6, and 5-HT7 receptors. Except...
    170 KB (17,955 words) - 12:34, 18 May 2025
  • Thumbnail for Receptor (biochemistry)
    In biochemistry and pharmacology, receptors are chemical structures, composed of protein, that receive and transduce signals that may be integrated into...
    26 KB (2,673 words) - 05:54, 5 May 2025
  • Thumbnail for HTR3B
    HTR3B (category Transmembrane receptor stubs)
    5-hydroxytryptamine (serotonin) receptor 3B, also known as HTR3B, is a human gene. The protein encoded by this gene is a subunit of the 5-HT3 receptor...
    8 KB (1,029 words) - 03:37, 29 November 2023
  • Thumbnail for Alpha-7 nicotinic receptor
    711: partial agonist Tropisetron: subtype-selective partial agonist; 5-HT3 receptor antagonist WAY-317,538 — selective potent full agonist with nootropic...
    28 KB (2,815 words) - 14:12, 9 May 2025
  • Thumbnail for Tropisetron
    Tropisetron (category 5-HT3 antagonists)
    Tropisetron is a serotonin 5-HT3 receptor antagonist used mainly as an antiemetic to treat nausea and vomiting following chemotherapy, although it has...
    7 KB (491 words) - 08:16, 14 January 2025
  • Thumbnail for Vortioxetine
    Vortioxetine (category 5-HT3 antagonists)
    the serotonin 5-HT1A receptor, partial agonist of the 5-HT1B receptor, and antagonist of the serotonin 5-HT1D, 5-HT3, and 5-HT7 receptors, as well as an...
    56 KB (4,812 words) - 17:40, 20 March 2025