• Thumbnail for Α5IA
    α5IA (LS-193,268) is a nootropic drug invented in 2004 by a team working for Merck, Sharp and Dohme, which acts as a subtype-selective inverse agonist...
    4 KB (281 words) - 23:16, 6 March 2024
  • Thumbnail for Α3IA
    subunits of the GABAA receptor, but it is more selective for the α3 subunit. α5IA, an inverse agonist at the α5 subunit of GABAA receptors "Alpha3IA". Atack...
    3 KB (194 words) - 19:58, 12 February 2024
  • Thumbnail for Penicillin
    Negative modulators: 1,3M1B 3M2B 11-Ketoprogesterone 17-Phenylandrostenol α3IA α5IA (LS-193,268) β-CCB β-CCE β-CCM β-CCP β-EMGBL Anabolic steroids Amiloride...
    97 KB (10,473 words) - 13:40, 15 April 2024
  • Thumbnail for GABAA receptor
    needed] Some of the subtype-selective negative allosteric modulators such as α5IA are being investigated for their nootropic effects, as well as treatments...
    54 KB (5,992 words) - 15:58, 28 March 2024
  • Thumbnail for Glutamine
    Negative modulators: 1,3M1B 3M2B 11-Ketoprogesterone 17-Phenylandrostenol α3IA α5IA (LS-193,268) β-CCB β-CCE β-CCM β-CCP β-EMGBL Anabolic steroids Amiloride...
    27 KB (2,443 words) - 08:45, 27 April 2024
  • Thumbnail for Gamma-Hydroxybutyric acid
    Negative modulators: 1,3M1B 3M2B 11-Ketoprogesterone 17-Phenylandrostenol α3IA α5IA (LS-193,268) β-CCB β-CCE β-CCM β-CCP β-EMGBL Anabolic steroids Amiloride...
    80 KB (8,754 words) - 18:02, 9 April 2024
  • Thumbnail for Ciprofloxacin
    Negative modulators: 1,3M1B 3M2B 11-Ketoprogesterone 17-Phenylandrostenol α3IA α5IA (LS-193,268) β-CCB β-CCE β-CCM β-CCP β-EMGBL Anabolic steroids Amiloride...
    66 KB (6,688 words) - 01:51, 21 April 2024
  • Thumbnail for Levofloxacin
    Negative modulators: 1,3M1B 3M2B 11-Ketoprogesterone 17-Phenylandrostenol α3IA α5IA (LS-193,268) β-CCB β-CCE β-CCM β-CCP β-EMGBL Anabolic steroids Amiloride...
    53 KB (5,404 words) - 01:47, 21 April 2024
  • Thumbnail for Lemon balm
    Negative modulators: 1,3M1B 3M2B 11-Ketoprogesterone 17-Phenylandrostenol α3IA α5IA (LS-193,268) β-CCB β-CCE β-CCM β-CCP β-EMGBL Anabolic steroids Amiloride...
    17 KB (1,632 words) - 16:10, 30 March 2024
  • Thumbnail for RDX
    Negative modulators: 1,3M1B 3M2B 11-Ketoprogesterone 17-Phenylandrostenol α3IA α5IA (LS-193,268) β-CCB β-CCE β-CCM β-CCP β-EMGBL Anabolic steroids Amiloride...
    57 KB (5,907 words) - 17:23, 6 March 2024
  • Thumbnail for Furosemide
    Negative modulators: 1,3M1B 3M2B 11-Ketoprogesterone 17-Phenylandrostenol α3IA α5IA (LS-193,268) β-CCB β-CCE β-CCM β-CCP β-EMGBL Anabolic steroids Amiloride...
    37 KB (3,648 words) - 20:31, 1 March 2024
  • Thumbnail for Γ-Aminobutyric acid
    Negative modulators: 1,3M1B 3M2B 11-Ketoprogesterone 17-Phenylandrostenol α3IA α5IA (LS-193,268) β-CCB β-CCE β-CCM β-CCP β-EMGBL Anabolic steroids Amiloride...
    51 KB (5,563 words) - 23:57, 21 March 2024
  • Thumbnail for Ofloxacin
    Negative modulators: 1,3M1B 3M2B 11-Ketoprogesterone 17-Phenylandrostenol α3IA α5IA (LS-193,268) β-CCB β-CCE β-CCM β-CCP β-EMGBL Anabolic steroids Amiloride...
    46 KB (4,449 words) - 16:10, 2 March 2024
  • Thumbnail for Phenibut
    Negative modulators: 1,3M1B 3M2B 11-Ketoprogesterone 17-Phenylandrostenol α3IA α5IA (LS-193,268) β-CCB β-CCE β-CCM β-CCP β-EMGBL Anabolic steroids Amiloride...
    31 KB (2,541 words) - 22:24, 17 April 2024
  • Negative modulators: 1,3M1B 3M2B 11-Ketoprogesterone 17-Phenylandrostenol α3IA α5IA (LS-193,268) β-CCB β-CCE β-CCM β-CCP β-EMGBL Anabolic steroids Amiloride...
    3 KB (315 words) - 21:55, 14 April 2024
  • Thumbnail for Flumazenil
    Negative modulators: 1,3M1B 3M2B 11-Ketoprogesterone 17-Phenylandrostenol α3IA α5IA (LS-193,268) β-CCB β-CCE β-CCM β-CCP β-EMGBL Anabolic steroids Amiloride...
    23 KB (2,416 words) - 16:54, 24 March 2024
  • Negative modulators: 1,3M1B 3M2B 11-Ketoprogesterone 17-Phenylandrostenol α3IA α5IA (LS-193,268) β-CCB β-CCE β-CCM β-CCP β-EMGBL Anabolic steroids Amiloride...
    2 KB (139 words) - 10:42, 29 October 2023
  • Thumbnail for 1,4-Butanediol
    Negative modulators: 1,3M1B 3M2B 11-Ketoprogesterone 17-Phenylandrostenol α3IA α5IA (LS-193,268) β-CCB β-CCE β-CCM β-CCP β-EMGBL Anabolic steroids Amiloride...
    18 KB (1,723 words) - 03:12, 9 April 2024
  • Thumbnail for Dehydroepiandrosterone
    Negative modulators: 1,3M1B 3M2B 11-Ketoprogesterone 17-Phenylandrostenol α3IA α5IA (LS-193,268) β-CCB β-CCE β-CCM β-CCP β-EMGBL Anabolic steroids Amiloride...
    42 KB (3,935 words) - 04:01, 30 April 2024
  • Thumbnail for Methylglyoxal
    Negative modulators: 1,3M1B 3M2B 11-Ketoprogesterone 17-Phenylandrostenol α3IA α5IA (LS-193,268) β-CCB β-CCE β-CCM β-CCP β-EMGBL Anabolic steroids Amiloride...
    13 KB (1,210 words) - 20:09, 10 March 2024
  • Thumbnail for Coriamyrtin
    Negative modulators: 1,3M1B 3M2B 11-Ketoprogesterone 17-Phenylandrostenol α3IA α5IA (LS-193,268) β-CCB β-CCE β-CCM β-CCP β-EMGBL Anabolic steroids Amiloride...
    4 KB (222 words) - 08:49, 21 February 2024
  • Thumbnail for Baclofen
    Negative modulators: 1,3M1B 3M2B 11-Ketoprogesterone 17-Phenylandrostenol α3IA α5IA (LS-193,268) β-CCB β-CCE β-CCM β-CCP β-EMGBL Anabolic steroids Amiloride...
    33 KB (3,204 words) - 00:31, 24 March 2024
  • Thumbnail for Muscimol
    Negative modulators: 1,3M1B 3M2B 11-Ketoprogesterone 17-Phenylandrostenol α3IA α5IA (LS-193,268) β-CCB β-CCE β-CCM β-CCP β-EMGBL Anabolic steroids Amiloride...
    26 KB (2,462 words) - 16:42, 28 April 2024
  • Thumbnail for Gamma-Butyrolactone
    Negative modulators: 1,3M1B 3M2B 11-Ketoprogesterone 17-Phenylandrostenol α3IA α5IA (LS-193,268) β-CCB β-CCE β-CCM β-CCP β-EMGBL Anabolic steroids Amiloride...
    29 KB (2,914 words) - 01:31, 27 March 2024
  • Thumbnail for Β-Carboline
    Negative modulators: 1,3M1B 3M2B 11-Ketoprogesterone 17-Phenylandrostenol α3IA α5IA (LS-193,268) β-CCB β-CCE β-CCM β-CCP β-EMGBL Anabolic steroids Amiloride...
    27 KB (2,633 words) - 08:14, 7 January 2024
  • Thumbnail for Isoflavonoid
    Negative modulators: 1,3M1B 3M2B 11-Ketoprogesterone 17-Phenylandrostenol α3IA α5IA (LS-193,268) β-CCB β-CCE β-CCM β-CCP β-EMGBL Anabolic steroids Amiloride...
    3 KB (242 words) - 16:07, 3 January 2024
  • Thumbnail for Lindane
    Negative modulators: 1,3M1B 3M2B 11-Ketoprogesterone 17-Phenylandrostenol α3IA α5IA (LS-193,268) β-CCB β-CCE β-CCM β-CCP β-EMGBL Anabolic steroids Amiloride...
    40 KB (4,019 words) - 18:12, 1 February 2024
  • Thumbnail for Thujone
    Negative modulators: 1,3M1B 3M2B 11-Ketoprogesterone 17-Phenylandrostenol α3IA α5IA (LS-193,268) β-CCB β-CCE β-CCM β-CCP β-EMGBL Anabolic steroids Amiloride...
    27 KB (2,621 words) - 01:26, 4 April 2024
  • Thumbnail for U-93631
    Negative modulators: 1,3M1B 3M2B 11-Ketoprogesterone 17-Phenylandrostenol α3IA α5IA (LS-193,268) β-CCB β-CCE β-CCM β-CCP β-EMGBL Anabolic steroids Amiloride...
    2 KB (126 words) - 01:21, 7 February 2024
  • Thumbnail for Phenytoin
    Negative modulators: 1,3M1B 3M2B 11-Ketoprogesterone 17-Phenylandrostenol α3IA α5IA (LS-193,268) β-CCB β-CCE β-CCM β-CCP β-EMGBL Anabolic steroids Amiloride...
    47 KB (4,510 words) - 19:00, 11 April 2024