• Thumbnail for Apalutamide
    Apalutamide, sold under the brand name Erleada among others, is a nonsteroidal antiandrogen (NSAA) medication which is used in the treatment of prostate...
    35 KB (3,082 words) - 23:02, 17 April 2024
  • impairment is unknown. Two 2020 meta-analyses reported that enzalutamide and apalutamide seemed to be more effective than darolutamide in improving metastasis-free...
    42 KB (4,163 words) - 09:13, 2 April 2024
  • Thumbnail for N-Desmethylapalutamide
    similar activity to that of apalutamide and, with apalutamide therapy, circulates at similar concentrations to those of apalutamide at steady state.[failed...
    3 KB (147 words) - 01:30, 8 August 2022
  • Thumbnail for Nonsteroidal antiandrogen
    Structurally distinct from enzalutamide, apalutamide, and other NSAAs. Relative to enzalutamide and apalutamide, shows greater efficacy as an AR antagonist...
    17 KB (1,576 words) - 15:57, 24 February 2024
  • ISSNĀ 0114-9954. S2CIDĀ 195107338. "Robust PSA Response and Treatment Adherence of Apalutamide in CRPC Seen with RWE". Targeted Oncology. 10 September 2021. Retrieved...
    25 KB (1,878 words) - 20:31, 23 April 2024
  • Thumbnail for Antiandrogen
    (also known as complete or maximal androgen blockade). Enzalutamide, apalutamide, and abiraterone acetate are specifically approved for use in combination...
    159 KB (15,186 words) - 12:25, 15 April 2024
  • Thumbnail for Glutamine
    MRK-016 Naloxone Naltrexone Nicardipine Nonsteroidal antiandrogens (e.g., apalutamide, bicalutamide, enzalutamide, flutamide, nilutamide) Oenanthotoxin Pentylenetetrazol...
    27 KB (2,492 words) - 16:02, 11 April 2024
  • Thumbnail for Testosterone
    acetate Oxendolone Potassium canrenoate Spironolactone Nonsteroidal: Apalutamide Bicalutamide Cimetidine Darolutamide Enzalutamide Flutamide Ketoconazole...
    149 KB (15,647 words) - 18:10, 15 April 2024
  • Thumbnail for List of antiandrogens
    First-generation Bicalutamide Flutamide Nilutamide Second-generation Apalutamide Darolutamide Enzalutamide Proxalutamide Others/non-generational Cimetidine...
    5 KB (254 words) - 18:23, 18 September 2023
  • Thumbnail for Ciprofloxacin
    MRK-016 Naloxone Naltrexone Nicardipine Nonsteroidal antiandrogens (e.g., apalutamide, bicalutamide, enzalutamide, flutamide, nilutamide) Oenanthotoxin Pentylenetetrazol...
    66 KB (6,688 words) - 01:51, 21 April 2024
  • Thumbnail for Phenibut
    MRK-016 Naloxone Naltrexone Nicardipine Nonsteroidal antiandrogens (e.g., apalutamide, bicalutamide, enzalutamide, flutamide, nilutamide) Oenanthotoxin Pentylenetetrazol...
    31 KB (2,541 words) - 22:24, 17 April 2024
  • Thumbnail for Furosemide
    MRK-016 Naloxone Naltrexone Nicardipine Nonsteroidal antiandrogens (e.g., apalutamide, bicalutamide, enzalutamide, flutamide, nilutamide) Oenanthotoxin Pentylenetetrazol...
    37 KB (3,648 words) - 20:31, 1 March 2024
  • Thumbnail for Trenbolone acetate
    acetate Oxendolone Potassium canrenoate Spironolactone Nonsteroidal: Apalutamide Bicalutamide Cimetidine Darolutamide Enzalutamide Flutamide Ketoconazole...
    33 KB (3,293 words) - 01:15, 23 February 2024
  • Thumbnail for Enzalutamide
    nilutamide, and bicalutamide as well as to newer second-generation NSAAs like apalutamide and proxalutamide. Enzalutamide was discovered by Charles Sawyers and...
    48 KB (4,545 words) - 06:42, 24 March 2024
  • Thumbnail for Stanozolol
    acetate Oxendolone Potassium canrenoate Spironolactone Nonsteroidal: Apalutamide Bicalutamide Cimetidine Darolutamide Enzalutamide Flutamide Ketoconazole...
    35 KB (3,320 words) - 17:12, 22 April 2024
  • Thumbnail for Gamma-Hydroxybutyric acid
    MRK-016 Naloxone Naltrexone Nicardipine Nonsteroidal antiandrogens (e.g., apalutamide, bicalutamide, enzalutamide, flutamide, nilutamide) Oenanthotoxin Pentylenetetrazol...
    80 KB (8,754 words) - 18:02, 9 April 2024
  • Thumbnail for Penicillin
    MRK-016 Naloxone Naltrexone Nicardipine Nonsteroidal antiandrogens (e.g., apalutamide, bicalutamide, enzalutamide, flutamide, nilutamide) Oenanthotoxin Pentylenetetrazol...
    97 KB (10,473 words) - 13:40, 15 April 2024
  • Thumbnail for Androgen
    acetate Oxendolone Potassium canrenoate Spironolactone Nonsteroidal: Apalutamide Bicalutamide Cimetidine Darolutamide Enzalutamide Flutamide Ketoconazole...
    29 KB (3,165 words) - 22:29, 23 March 2024
  • Thumbnail for Baclofen
    MRK-016 Naloxone Naltrexone Nicardipine Nonsteroidal antiandrogens (e.g., apalutamide, bicalutamide, enzalutamide, flutamide, nilutamide) Oenanthotoxin Pentylenetetrazol...
    33 KB (3,204 words) - 00:31, 24 March 2024
  • Thumbnail for Azelaic acid
    (R-2956) Zanoterone Nonsteroidal: 5N-Bicalutamide AA560 Antarlides Arabilin Apalutamide Atraric acid AZD-3514 Bakuchiol Bavdegalutamide BAY-1024767 Bicalutamide...
    17 KB (1,611 words) - 18:36, 5 January 2024
  • Thumbnail for Prostate cancer
    antiandrogen drugs, namely the androgen receptor antagonists enzalutamide, apalutamide, and darolutamide, as well as the testosterone production inhibitor abiraterone...
    77 KB (8,858 words) - 14:12, 23 April 2024
  • Thumbnail for Levofloxacin
    MRK-016 Naloxone Naltrexone Nicardipine Nonsteroidal antiandrogens (e.g., apalutamide, bicalutamide, enzalutamide, flutamide, nilutamide) Oenanthotoxin Pentylenetetrazol...
    53 KB (5,404 words) - 01:47, 21 April 2024
  • Thumbnail for Trenbolone
    acetate Oxendolone Potassium canrenoate Spironolactone Nonsteroidal: Apalutamide Bicalutamide Cimetidine Darolutamide Enzalutamide Flutamide Ketoconazole...
    18 KB (1,331 words) - 16:47, 13 April 2024
  • Thumbnail for RDX
    MRK-016 Naloxone Naltrexone Nicardipine Nonsteroidal antiandrogens (e.g., apalutamide, bicalutamide, enzalutamide, flutamide, nilutamide) Oenanthotoxin Pentylenetetrazol...
    57 KB (5,907 words) - 17:23, 6 March 2024
  • Thumbnail for Testosterone propionate/testosterone phenylpropionate/testosterone isocaproate/testosterone decanoate
    acetate Oxendolone Potassium canrenoate Spironolactone Nonsteroidal: Apalutamide Bicalutamide Cimetidine Darolutamide Enzalutamide Flutamide Ketoconazole...
    7 KB (383 words) - 20:10, 20 December 2023
  • Thumbnail for Mifepristone
    (R-2956) Zanoterone Nonsteroidal: 5N-Bicalutamide AA560 Antarlides Arabilin Apalutamide Atraric acid AZD-3514 Bakuchiol Bavdegalutamide BAY-1024767 Bicalutamide...
    119 KB (11,038 words) - 18:04, 15 April 2024
  • Thumbnail for Oxandrolone
    acetate Oxendolone Potassium canrenoate Spironolactone Nonsteroidal: Apalutamide Bicalutamide Cimetidine Darolutamide Enzalutamide Flutamide Ketoconazole...
    47 KB (4,508 words) - 12:16, 22 April 2024
  • MRK-016 Naloxone Naltrexone Nicardipine Nonsteroidal antiandrogens (e.g., apalutamide, bicalutamide, enzalutamide, flutamide, nilutamide) Oenanthotoxin Pentylenetetrazol...
    2 KB (139 words) - 10:42, 29 October 2023
  • Thumbnail for Ketoconazole
    acetate Oxendolone Potassium canrenoate Spironolactone Nonsteroidal: Apalutamide Bicalutamide Cimetidine Darolutamide Enzalutamide Flutamide Ketoconazole...
    50 KB (4,369 words) - 10:03, 6 April 2024
  • Thumbnail for Coriamyrtin
    MRK-016 Naloxone Naltrexone Nicardipine Nonsteroidal antiandrogens (e.g., apalutamide, bicalutamide, enzalutamide, flutamide, nilutamide) Oenanthotoxin Pentylenetetrazol...
    4 KB (222 words) - 08:49, 21 February 2024