• Thumbnail for Bicuculline
    Bicuculline is a phthalide-isoquinoline compound that is a light-sensitive competitive antagonist of GABAA receptors. It was originally identified in...
    5 KB (316 words) - 20:39, 11 April 2024
  • Thumbnail for GABA receptor
    It has long been recognized that, for neurons that are stimulated by bicuculline and picrotoxin, the fast inhibitory response to GABA is due to direct...
    35 KB (3,884 words) - 20:11, 11 February 2024
  • used for counteracting overdoses of sedative drugs. Examples include bicuculline, securinine and metrazol, and the benzodiazepine GABAA receptor antagonist...
    3 KB (315 words) - 21:55, 14 April 2024
  • endogenous and exogenous actions of GABAA receptor agonists. Bemegride Bicuculline Cicutoxin Cyclothiazide DMCM FG-7142 Fipronil Flumazenil Flurothyl Gabazine...
    13 KB (1,191 words) - 17:00, 18 February 2024
  • Thumbnail for Glycine
    Strychnine is a strong antagonist at ionotropic glycine receptors, whereas bicuculline is a weak one. Glycine is a required co-agonist along with glutamate...
    37 KB (3,313 words) - 15:36, 19 March 2024
  • Thumbnail for Cocaine
    TC-2216 Tebanicline UB-165 Varenicline WAY-317,538 Convulsants Anatoxin-a Bicuculline DMCM Flurothyl Gabazine Pentetrazol Picrotoxin Strychnine Thujone Eugeroics...
    161 KB (17,714 words) - 21:10, 9 April 2024
  • PMID 21833169. Hill DR, Bowery NG (March 1981). "3H-baclofen and 3H-GABA bind to bicuculline-insensitive GABA B sites in rat brain". Nature. 290 (5802): 149–52. Bibcode:1981Natur...
    16 KB (1,564 words) - 20:19, 25 March 2024
  • Thumbnail for MDMA
    TC-2216 Tebanicline UB-165 Varenicline WAY-317,538 Convulsants Anatoxin-a Bicuculline DMCM Flurothyl Gabazine Pentetrazol Picrotoxin Strychnine Thujone Eugeroics...
    151 KB (15,039 words) - 15:18, 12 April 2024
  • Thumbnail for Alcohol (drug)
    2-Aminostrychnine 2-Nitrostrychnine 4-Phenyl-4-formyl-N-methylpiperidine αEMBTL Bicuculline Brucine Cacotheline Caffeine Colchicine Colubrine Cyanotriphenylborate...
    185 KB (18,571 words) - 00:07, 16 April 2024
  • 2-Aminostrychnine 2-Nitrostrychnine 4-Phenyl-4-formyl-N-methylpiperidine αEMBTL Bicuculline Brucine Cacotheline Caffeine Colchicine Colubrine Cyanotriphenylborate...
    21 KB (1,924 words) - 21:51, 11 April 2024
  • Thumbnail for Methamphetamine
    TC-2216 Tebanicline UB-165 Varenicline WAY-317,538 Convulsants Anatoxin-a Bicuculline DMCM Flurothyl Gabazine Pentetrazol Picrotoxin Strychnine Thujone Eugeroics...
    150 KB (14,825 words) - 20:44, 11 March 2024
  • Thumbnail for Gabazine
    Heinemann U (April 2007). "Effects of the GABA(A) receptor antagonists bicuculline and gabazine on stimulus-induced sharp wave-ripple complexes in adult...
    4 KB (324 words) - 04:35, 25 March 2024
  • Thumbnail for Flunitrazepam
    2-Aminostrychnine 2-Nitrostrychnine 4-Phenyl-4-formyl-N-methylpiperidine αEMBTL Bicuculline Brucine Cacotheline Caffeine Colchicine Colubrine Cyanotriphenylborate...
    38 KB (3,691 words) - 21:44, 15 March 2024
  • Thumbnail for Muscimol
    Woodward RM, Polenzani L, Miledi R (April 1993). "Characterization of bicuculline/baclofen-insensitive (rho-like) gamma-aminobutyric acid receptors expressed...
    26 KB (2,462 words) - 12:17, 23 March 2024
  • Thumbnail for Morphine
    2-Aminostrychnine 2-Nitrostrychnine 4-Phenyl-4-formyl-N-methylpiperidine αEMBTL Bicuculline Brucine Cacotheline Caffeine Colchicine Colubrine Cyanotriphenylborate...
    140 KB (13,643 words) - 04:49, 9 April 2024
  • Thumbnail for ROD-188
    was structurally derived from the GABAA antagonist bicuculline by a team at Roche. Unlike bicuculline, ROD-188 acts as an agonist at GABAA receptors, being...
    3 KB (239 words) - 18:33, 12 August 2023
  • Thumbnail for Phencyclidine
    TC-2216 Tebanicline UB-165 Varenicline WAY-317,538 Convulsants Anatoxin-a Bicuculline DMCM Flurothyl Gabazine Pentetrazol Picrotoxin Strychnine Thujone Eugeroics...
    55 KB (5,314 words) - 00:33, 3 April 2024
  • Thumbnail for Barbiturate
    2-Aminostrychnine 2-Nitrostrychnine 4-Phenyl-4-formyl-N-methylpiperidine αEMBTL Bicuculline Brucine Cacotheline Caffeine Colchicine Colubrine Cyanotriphenylborate...
    44 KB (4,697 words) - 15:28, 5 April 2024
  • Thumbnail for Adderall
    TC-2216 Tebanicline UB-165 Varenicline WAY-317,538 Convulsants Anatoxin-a Bicuculline DMCM Flurothyl Gabazine Pentetrazol Picrotoxin Strychnine Thujone Eugeroics...
    56 KB (19,815 words) - 10:12, 28 February 2024
  • Thumbnail for Psychoactive drug
    receptor positive allosteric modulators GABA receptor antagonists thujone, bicuculline GABAA receptor negative allosteric modulators Norepinephrine Norepinephrine...
    64 KB (6,249 words) - 18:12, 9 April 2024
  • Thumbnail for GABAA receptor
    binding site for GABA and several drugs such as muscimol, gaboxadol, and bicuculline. The protein also contains a number of different allosteric binding sites...
    54 KB (5,992 words) - 15:58, 28 March 2024
  • Thumbnail for Diethyl ether
    2-Aminostrychnine 2-Nitrostrychnine 4-Phenyl-4-formyl-N-methylpiperidine αEMBTL Bicuculline Brucine Cacotheline Caffeine Colchicine Colubrine Cyanotriphenylborate...
    28 KB (2,743 words) - 08:14, 5 April 2024
  • Thumbnail for Γ-Aminobutyric acid
    Ueno, S; Bracamontes, J; Zorumski, C; Weiss, DS; Steinbach, JH (1997). "Bicuculline and gabazine are allosteric inhibitors of channel opening of the GABAA...
    51 KB (5,563 words) - 23:57, 21 March 2024
  • Thumbnail for Nefiracetam
    impairing substances, including: ethanol, chlorodiazepoxide, scopolamine, bicuculline, picrotoxin, and cycloheximide. Unlike other racetams, nefiracetam shows...
    8 KB (732 words) - 06:00, 7 September 2023
  • Thumbnail for Stimulant
    TC-2216 Tebanicline UB-165 Varenicline WAY-317,538 Convulsants Anatoxin-a Bicuculline DMCM Flurothyl Gabazine Pentetrazol Picrotoxin Strychnine Thujone Eugeroics...
    125 KB (13,051 words) - 19:54, 14 April 2024
  • Thumbnail for Caffeine
    TC-2216 Tebanicline UB-165 Varenicline WAY-317,538 Convulsants Anatoxin-a Bicuculline DMCM Flurothyl Gabazine Pentetrazol Picrotoxin Strychnine Thujone Eugeroics...
    197 KB (19,765 words) - 21:10, 11 April 2024
  • Thumbnail for Alcoholism
    interoceptive stimulus produced by ethanol withdrawal is potentiated by bicuculline and picrotoxinin". Neuropsychopharmacology. 2 (2): 115–22. doi:10...
    141 KB (14,394 words) - 07:04, 12 March 2024
  • Thumbnail for Glutamine
    hydrate, chloroform, diethyl ether, paraldehyde, sevoflurane) Antagonists: Bicuculline Coriamyrtin Dihydrosecurinine Gabazine (SR-95531) Hydrastine Hyenachin...
    27 KB (2,492 words) - 16:02, 11 April 2024
  • the blood brain barrier and enter the brain Bicuculline methiodide, a water-soluble form of bicuculline Tertiary phosphines and phosphite esters also...
    1 KB (162 words) - 13:59, 22 April 2022
  • Thumbnail for Alcohol withdrawal syndrome
    interoceptive stimulus produced by ethanol withdrawal is potentiated by bicuculline and picrotoxinin". Neuropsychopharmacology. 2 (2): 115–22. doi:10...
    41 KB (4,124 words) - 11:04, 7 April 2024