The cannabinoid receptor 2 (CB2), is a G protein-coupled receptor from the cannabinoid receptor family that in humans is encoded by the CNR2 gene. It...

Cannabinoid receptors, located throughout the body, are part of the endocannabinoid system of vertebrates– a class of cell membrane receptors in the G...

A cannabinoid receptor antagonist, also known simply as a cannabinoid antagonist or as an anticannabinoid, is a type of cannabinoidergic drug that binds...

Cannabinoid receptor 1 (CB1), is a G protein-coupled cannabinoid receptor that in humans is encoded by the CNR1 gene. The human CB1 receptor is expressed...

animal organisms (although insects lack such receptors) or as synthetic compounds. The most notable cannabinoid is the phytocannabinoid tetrahydrocannabinol...

lipid-based retrograde neurotransmitters that bind to cannabinoid receptors, and cannabinoid receptor proteins that are expressed throughout the vertebrate...

Synthetic cannabinoids are a class of designer drug molecules that bind to the same receptors to which cannabinoids (THC, CBD and many others) in cannabis...

1999). "Evidence that the cannabinoid CB1 receptor is a 2-arachidonoylglycerol receptor. Structure-activity relationship of 2-arachidonoylglycerol, ether-linked...

dose-dependent buildup of cannabinoids and related effects of cannabinoid toxicity the functionality of cannabinoid receptors in the brain and particularly...

vasopressin receptor 2 β-adrenergic receptors types β1, β2 and β3 Calcitonin receptor Calcitonin gene-related peptide receptor Cannabinoid receptor 2 Corticotropin-releasing...

has an entirely different chemical structure. WIN 55,212-2 is a potent cannabinoid receptor agonist that has been found to be a potent analgesic in a...

(ACPA) is a synthetic agonist of the cannabinoid receptor 1 (CB1R). ACPA is considered to be a selective cannabinoid agonist as it binds primarily to the...

protein-coupled receptors (GPCRs), also known as seven-(pass)-transmembrane domain receptors, 7TM receptors, heptahelical receptors, serpentine receptors, and G...

receptors Adrenergic α2A, α2B, & α2C receptors Apelin receptors Calcium-sensing receptor Cannabinoid receptors (CB1 and CB2) Chemokine CXCR4 receptor...

is the compound's binding affinity for the cannabinoid receptor type 1 (CB1) or cannabinoid receptor type 2 (CB2). Manera C, Tuccinardi T, Martinelli A...

CB2 cannabinoid receptors, with some selectivity for CB2. It produces effects in animals similar to those of tetrahydrocannabinol (THC), a cannabinoid naturally...

389–462. doi:10.1124/pr.58.3.2. PMC 2241751. PMID 16968947. Hongfeng Deng. Design and synthesis of selective cannabinoid receptor ligands: Aminoalkylindole...

etonitazene itself. This compound was also tested as part of a series of cannabinoid receptor 2 agonists, and was found to be active though with fairly low potency...

potent but nonselective full agonist for the cannabinoid receptor. It is part of the AM series of cannabinoids discovered by Alexandros Makriyannis at Northeastern...

agonist at the CB1 cannabinoid receptor. AM-251 is structurally very close to rimonabant; both are biarylpyrazole cannabinoid receptor antagonists. In AM-251...

GPR55, along with GPR119 and GPR18, have been implicated as novel cannabinoid receptors. GPR55 was identified and cloned for the first time in 1999. Later...

The beta-2 adrenergic receptor (β2 adrenoreceptor), also known as ADRB2, is a cell membrane-spanning beta-adrenergic receptor that binds epinephrine (adrenaline)...

inverse agonist for the cannabinoid receptor CB1 and was first-in-class for clinical development. Rimonabant is a selective CB1 receptor blocker and was discovered...

functions differently in rat cannabinoid receptors binding to rat cannabinoid CB2 receptors at Ki = 16.3 ± 2.1 and CB1 receptors at Ki = 1130 ± 574 nM binding...

The alpha-2 (α2) adrenergic receptor (or adrenoceptor) is a G protein-coupled receptor (GPCR) associated with the Gi heterotrimeric G-protein. It consists...

(also incorrectly known as 5-CL-ADB-A) is an indazole-based synthetic cannabinoid that has been sold online as a designer drug. MDMB-4en-PINACA was first...

AM-679 (part of the AM cannabinoid series) is a drug that acts as a moderately potent agonist for the cannabinoid receptors, with a Ki of 13.5 nM at CB1...

receptor (PTAFR, PAFR) InterPro: IPR002282 Cannabinoid receptor InterPro: IPR002230 Cannabinoid receptor 1 (brain) (CNR1, CB1R) Cannabinoid receptor 2...

Zhang M, Tuma R, Son YJ, Persidsky Y (March 2012). "Activation of cannabinoid receptor 2 attenuates leukocyte-endothelial cell interactions and blood-brain...

Michelle; Graham, Euan Scott; Grimsey, Natasha Lillia (2019-10-19). "Cannabinoid Receptor 2 (CB 2 ) Signals via G-alpha-s and Induces IL-6 and IL-10 Cytokine Secretion...