Dopamine receptor D5, also known as D1BR, is a protein that in humans is encoded by the DRD5 gene. It belongs to the D1-like receptor family along with... 37 KB (4,376 words) - 23:19, 9 February 2024 |
Dopamine receptor D1, also known as DRD1. It is one of the two types of D1-like receptor family — receptors D1 and D5. It is a protein that in humans... 31 KB (3,089 words) - 23:16, 9 February 2024 |
dopamine antagonist, also known as an anti-dopaminergic and a dopamine receptor antagonist (DRA), is a type of drug which blocks dopamine receptors by... 31 KB (3,140 words) - 02:58, 26 March 2024 |
Dopamine receptor D2, also known as D2R, is a protein that, in humans, is encoded by the DRD2 gene. After work from Paul Greengard's lab had suggested... 34 KB (3,958 words) - 20:55, 28 March 2024 |
The dopamine receptor D4 is a dopamine D2-like G protein-coupled receptor encoded by the DRD4 gene on chromosome 11 at 11p15.5. The structure of DRD4... 36 KB (4,060 words) - 01:53, 4 April 2024 |
Dopamine receptor D3 is a protein that in humans is encoded by the DRD3 gene. This gene encodes the D3 subtype of the dopamine receptor. The D3 subtype... 28 KB (3,175 words) - 04:10, 4 January 2024 |
The D1-like receptors are a subfamily of dopamine receptors that bind the endogenous neurotransmitter dopamine. The D1-like subfamily consists of two G... 2 KB (140 words) - 08:43, 3 January 2023 |
Tavapadon (category D5 receptor agonists) 2018. It acts as a selective partial agonist of the dopamine D1 (Ki = 8.54 nM) and D5 receptors. It also shows biased agonism for Gs-coupled signaling... 4 KB (169 words) - 01:58, 11 February 2024 |
Rotigotine (category D5 receptor agonists) non-selective agonist of the dopamine D1, D2, D3, and, to a lesser extent, D4 and D5 receptors, with highest affinity for the D3 receptor. In terms of affinity... 13 KB (1,068 words) - 11:46, 13 April 2024 |
South Western Motorway, Sydney, Australia Vitamin D5 D5, also known as DRD5, a subtype of dopamine receptors A 5% dextrose solution, a type of intravenous... 2 KB (239 words) - 12:49, 11 September 2023 |
response to the activity-initiated calcium influx. Activation of dopamine receptor D5 also promotes expression of BDNF in prefrontal cortex neurons. BDNF... 45 KB (5,339 words) - 00:15, 22 March 2024 |
Dihydrexidine (category D5 receptor agonists) selective full agonist at the dopamine D1 and D5 receptors. It has approximately 10-fold selectivity for D1 and D5 over the D2 receptor. Although dihydrexidine... 7 KB (647 words) - 02:22, 26 July 2023 |
SKF-81,297 (category D5 receptor agonists) drug of the benzazepine chemical class that acts as a selective dopamine D1/D5 receptor full agonist, and produces a characteristic stimulant-like pattern... 4 KB (398 words) - 11:21, 12 February 2023 |
(July 2001). "kappa-Opioid receptor agonist-induced prolactin release in primates is blocked by dopamine D(2)-like receptor agonists". European Journal... 67 KB (7,675 words) - 03:40, 2 May 2024 |
body. These two receptors also have important roles in the brain, regulating the release of other neurotransmitters such as dopamine and glutamate, while... 20 KB (1,954 words) - 16:46, 22 April 2024 |
if dopamine is safe to use during pregnancy or breastfeeding. At low doses dopamine mainly triggers dopamine receptors and β1-adrenergic receptors while... 17 KB (1,316 words) - 18:26, 24 March 2024 |
Ecopipam (category Dopamine antagonists) syndrome. It is taken by mouth. Ecopipam acts as a selective dopamine D1 and D5 receptor antagonist. It is orally active, has an elimination half-life... 14 KB (1,375 words) - 16:31, 24 March 2024 |
the treatment of anxiety and depression. 5-HT1A receptor activation has been shown to increase dopamine release in the medial prefrontal cortex, striatum... 58 KB (6,122 words) - 04:02, 3 May 2024 |
The alpha-2 (α2) adrenergic receptor (or adrenoceptor) is a G protein-coupled receptor (GPCR) associated with the Gi heterotrimeric G-protein. It consists... 25 KB (2,226 words) - 23:08, 28 April 2024 |
SKF-38,393 (category D5 receptor agonists) compound of the benzazepine chemical class which acts as a selective D1/D5 receptor partial agonist. It has stimulant and anorectic effects. The trimethylation... 3 KB (197 words) - 04:10, 30 March 2024 |