• Thumbnail for Estradiol sulfamate
    Estradiol sulfamate (E2MATE; developmental code names J995, PGL-2, PGL-2001, ZK-190628, others), or estradiol-3-O-sulfamate, is a steroid sulfatase (STS)...
    16 KB (1,643 words) - 11:10, 15 January 2024
  • Thumbnail for Pharmacokinetics of estradiol
    The pharmacology of estradiol, an estrogen medication and naturally occurring steroid hormone, concerns its pharmacodynamics, pharmacokinetics, and various...
    223 KB (26,822 words) - 02:01, 1 May 2024
  • Thumbnail for List of estrogen esters
    glucuronide Estradiol linoleate Estradiol oleate Estradiol phosphate Estradiol salicylate (estradiol 3-salicylate) Estradiol sulfamate (E2MATE; J995, PGL-2, PGL-2001...
    21 KB (2,022 words) - 18:43, 3 December 2023
  • Thumbnail for Estradiol
    Estradiol (E2), also spelled oestradiol, is an estrogen steroid hormone and the major female sex hormone. It is involved in the regulation of female reproductive...
    72 KB (7,059 words) - 16:31, 11 May 2024
  • Thumbnail for Estradiol (medication)
    Estradiol (E2) is a medication and naturally occurring steroid hormone. It is an estrogen and is used mainly in menopausal hormone therapy and to treat...
    162 KB (15,421 words) - 05:52, 8 April 2024
  • Thumbnail for Estradiol valerate
    Estradiol valerate (EV), sold for use by mouth under the brand name Progynova and for use by injection under the brand names Delestrogen and Progynon...
    86 KB (9,431 words) - 23:55, 18 March 2024
  • Thumbnail for Estradiol disulfate
    Estradiol disulfate (also known as E2DS or estradiol 3,17β-disulfate) is an endogenous estrogen conjugate and metabolite of estradiol. It is related to...
    3 KB (159 words) - 20:26, 8 November 2022
  • Instead, other non-oral forms of estradiol such as transdermal estradiol are recommended and may be used. Estradiol injectables are generally well-tolerated...
    111 KB (12,428 words) - 06:16, 11 March 2024
  • Thumbnail for Estradiol enantate
    Estradiol enantate (EEn or E2-EN), also spelled estradiol enanthate and sold under the brand names Perlutal and Topasel among others, is an estrogen medication...
    55 KB (4,716 words) - 08:37, 10 March 2024
  • Thumbnail for Estrogen
    that have estrogenic hormonal activity: estrone (E1), estradiol (E2), and estriol (E3). Estradiol, an estrane, is the most potent and prevalent. Another...
    72 KB (7,575 words) - 07:57, 13 April 2024
  • women include estradiol, which is the predominant natural estrogen in women, and estradiol esters such as estradiol valerate and estradiol cypionate, which...
    229 KB (24,526 words) - 03:11, 10 May 2024
  • sulfate), sulfamic acid (as in estradiol sulfamate), phosphoric acid (as in estradiol phosphate), glucuronic acid (as in estradiol glucuronide, and others (e...
    21 KB (2,080 words) - 23:33, 8 December 2023
  • Thumbnail for Estriol sulfamate
    hepatic estrogenic potency. However, the closely related compound estradiol sulfamate (E2MATE) failed to show estrogenic activity in humans, which is due...
    5 KB (368 words) - 14:39, 24 October 2023
  • Thumbnail for Estrone sulfamate
    an effective prodrug of estrogens. A closely related compound is estradiol sulfamate (E2MATE), which is extensively metabolized into EMATE and has similar...
    8 KB (683 words) - 15:07, 29 December 2023
  • Thumbnail for Estradiol benzoate
    Estradiol benzoate (EB), sold under the brand name Progynon-B among others, is an estrogen medication which is used in hormone therapy for menopausal...
    67 KB (6,903 words) - 16:31, 11 May 2024
  • Thumbnail for Estradiol furoate
    Estradiol furoate (EF), or estradiol 17β-furoate, sold under the brand name Di-Folliculine, is an estrogen medication and estrogen ester which is no longer...
    4 KB (188 words) - 20:27, 8 November 2022
  • Thumbnail for EC508
    properties and the mechanism by which they occur. Estradiol sulfamate (E2MATE) is a C3 sulfamate ester of estradiol which was developed in the 1990s and was a...
    15 KB (1,349 words) - 23:59, 10 May 2024
  • Thumbnail for Ethinylestradiol sulfamate
    similar properties in animals. However, the closely related compound estradiol sulfamate (E2MATE) failed to show estrogenic activity in humans, which is due...
    6 KB (356 words) - 18:43, 3 December 2023
  • Thumbnail for Estradiol cypionate
    Estradiol cypionate (EC), sold under the brand name Depo-Estradiol among others, is an estrogen medication which is used in hormone therapy for menopausal...
    51 KB (5,105 words) - 19:48, 9 May 2024
  • Thumbnail for Estradiol undecylate
    Estradiol undecylate (EU, EUn, E2U), also known as estradiol undecanoate and formerly sold under the brand names Delestrec and Progynon Depot 100 among...
    82 KB (7,980 words) - 03:44, 3 May 2024
  • Thumbnail for Estradiol pivalate
    Estradiol pivalate, also known as estradiol trimethyl acetate (E2-TMA) and sold under the brand name Estrotate, is an estrogen medication and an estrogen...
    9 KB (700 words) - 23:04, 19 March 2024
  • Thumbnail for Estrogen (medication)
    routes of administration. Examples of estrogens include bioidentical estradiol, natural conjugated estrogens, synthetic steroidal estrogens like ethinylestradiol...
    131 KB (14,549 words) - 07:58, 13 April 2024
  • The pharmacology of estradiol, an estrogen medication and naturally occurring steroid hormone, concerns its pharmacodynamics, pharmacokinetics, and various...
    103 KB (12,043 words) - 18:30, 24 March 2024
  • Thumbnail for Conjugated estrogens
    estrogen receptor, the biological target of estrogens like estradiol. Compared to estradiol, certain estrogens in CEEs are more resistant to metabolism...
    58 KB (6,452 words) - 05:22, 30 April 2024
  • This is a list of currently marketed formulations of estradiol benzoate (EB) throughout the world. Both EB alone and combinations of EB with other medications...
    7 KB (596 words) - 21:01, 11 November 2023
  • neurosteroids. Steroid sulfatase (STS) inhibitors such as estradiol sulfamate, estrone sulfamate, irosustat, and danazol inhibit the conversion of steroid...
    37 KB (2,107 words) - 11:12, 27 September 2022
  • Thumbnail for Estramustine phosphate
    Estramustine phosphate (category Estradiol esters)
    Estramustine phosphate (EMP), also known as estradiol normustine phosphate and sold under the brand names Emcyt and Estracyt, is a dual estrogen and chemotherapy...
    69 KB (6,639 words) - 19:57, 20 December 2023
  • control pills that contain natural estradiol or an estradiol ester (e.g., estradiol valerate) include: Estradiol valerate and cyproterone acetate (brand...
    9 KB (876 words) - 04:41, 30 August 2023
  • Thumbnail for Ethinylestradiol sulfonate
    to the development of estrogen sulfamates like estradiol 3-sulfamate (J995), estriol 3-sulfamate (J1034), and estradiol 17β-(1-(4-(aminosulfonyl)benzoyl)-L-proline)...
    24 KB (2,279 words) - 00:34, 9 December 2023
  • Thumbnail for Steroid sulfatase
    irosustat, estrone sulfamate (EMATE), estradiol sulfamate (E2MATE), and danazol. The most potent inhibitors are based around the aryl sulfamate pharmacophore...
    19 KB (2,144 words) - 04:03, 10 May 2024