Ionotropic GABA receptors (iGABARs) are ligand-gated ion channel of the GABA receptors class which are activated by gamma-aminobutyric acid (GABA), and... 7 KB (687 words) - 19:31, 11 February 2023 |
γ subunits of GABA receptors to improve GABAergic signaling. Alcohol also modulates ionotropic GABA receptors. Metabotropic receptors are often G-protein-coupled... 22 KB (2,705 words) - 08:12, 8 January 2024 |
transmission. GABA calms the brain and controls several physiological processes, such as stress, anxiety, and sleep. GABAA receptors are a class of ionotropic receptors... 11 KB (1,274 words) - 21:20, 19 February 2024 |
Molecular neuroscience (section Ionotropic receptors) generated by lower GABA concentrations. Ionotropic glutamate receptors can include NMDA, AMPA, and kainate receptors. These receptors are named after agonists... 26 KB (3,050 words) - 14:32, 10 September 2021 |
muscle relaxant effects. There are three receptors of the gamma-aminobutyric acid. The two receptors GABA-α and GABA-ρ are ion channels that are permeable... 8 KB (740 words) - 19:39, 11 March 2024 |
An ionotropic effect is the effect of a transmitter substance or hormone that activates or deactivates ionotropic receptors (ligand-gated ion channels)... 1 KB (96 words) - 06:14, 27 December 2023 |
Ligand-gated ion channel (redirect from Ionotropic receptors) Ligand-gated ion channels (LICs, LGIC), also commonly referred to as ionotropic receptors, are a group of transmembrane ion-channel proteins which open to... 30 KB (2,597 words) - 04:19, 25 March 2024 |
Γ-Aminobutyric acid (redirect from Gaba agents) metabotropic receptors, which are G protein-coupled receptors that open or close ion channels via intermediaries (G proteins) Neurons that produce GABA as their... 51 KB (5,563 words) - 23:57, 21 March 2024 |
Kainate receptors, or kainic acid receptors (KARs), are ionotropic receptors that respond to the neurotransmitter glutamate. They were first identified... 11 KB (1,264 words) - 23:19, 4 March 2024 |
to other GABAA receptors, the GABAA-ρ receptor has especially high expression in the retina. A second type of ionotropic GABA receptor, insensitive to... 16 KB (1,639 words) - 05:16, 7 November 2023 |
The glycine receptor (abbreviated as GlyR or GLR) is the receptor of the amino acid neurotransmitter glycine. GlyR is an ionotropic receptor that produces... 14 KB (1,546 words) - 19:55, 4 March 2024 |
(or inverse agonists) at either the GABAA or glycine receptors, or ionotropic glutamate receptor agonists. Many other drugs may cause convulsions as a... 13 KB (1,191 words) - 17:00, 18 February 2024 |
Gamma-Amino-beta-hydroxybutyric acid (redirect from Β-hydroxy-GABA) anticonvulsant and is used in the treatment of epilepsy. GABOB is a GABA receptor agonist. It has two stereoisomers, and shows stereoselectivity in its... 8 KB (688 words) - 09:14, 5 December 2023 |
Muscimol (category GABAA receptor agonists) ncbi.nlm.nih.gov. Johnston GA (October 2014). "Muscimol as an ionotropic GABA receptor agonist". Neurochemical Research. 39 (10): 1942–1947. doi:10... 26 KB (2,462 words) - 12:17, 23 March 2024 |
Phenibut (redirect from Phenyl-GABA) neurotransmitter γ-aminobutyric acid (GABA), and hence is a GABA analogue. Phenibut is thought to act as a GABAB receptor agonist, similarly to baclofen and... 31 KB (2,537 words) - 16:24, 21 March 2024 |
Thujone (category GABAA receptor negative allosteric modulators) neuropharm.2003.09.022. PMID 15002407. S2CID 54346490. Modulation of Ionotropic GABA Receptors by Natural Products of Plant Origin Naser B, Bodinet C, Tegtmeier... 27 KB (2,630 words) - 20:59, 21 March 2024 |
Neurotransmitter (redirect from Receptors, neurotransmitter) interact with receptors on the target cell. The effect of the neurotransmitter is dependent on the identity of the target cell's receptors present at the... 94 KB (8,335 words) - 06:00, 26 February 2024 |
4-Fluorophenibut (redirect from Β-(4-fluorophenyl)-GABA) β-(4-fluorophenyl)-GABA) is a GABAB receptor agonist which was never marketed. It is selective for the GABAB receptor over the GABAA receptor (IC50 = 1.70 μM... 4 KB (193 words) - 16:16, 21 March 2024 |
Theories of general anaesthetic action (section GABAA receptor is a major target of general anesthetics) Letourneur, Diane; Legendre, Pascal (2021). "Electrophysiology of ionotropic GABA receptors". Cellular and Molecular Life Sciences. 78 (13): 5341–5370. doi:10... 62 KB (6,743 words) - 16:45, 24 March 2024 |