A serotonin antagonist, or serotonin receptor antagonist, is a drug used to inhibit the action of serotonin and serotonergic drugs at serotonin (5-HT)... 5 KB (506 words) - 03:46, 13 August 2023 |
5-HT receptors, 5-hydroxytryptamine receptors, or serotonin receptors, are a group of G protein-coupled receptor and ligand-gated ion channels found in... 65 KB (5,263 words) - 05:49, 28 March 2024 |
fit into this class as it does not function as a serotonin antagonist, acting solely as a 5-HT1A receptor partial agonist instead. Vortioxetine (Trintellix)... 9 KB (615 words) - 21:41, 9 March 2024 |
A serotonin receptor agonist is an agonist of one or more serotonin receptors. They activate serotonin receptors in a manner similar to that of serotonin... 16 KB (1,657 words) - 23:51, 26 May 2023 |
which acts as a serotonin reuptake inhibitor (SRI), agonist of the 5-HT1A receptor, and antagonist of the 5-HT3 and 5-HT7 receptors. However, it can... 5 KB (568 words) - 17:03, 21 March 2024 |
A vasopressin receptor antagonist (VRA) is an agent that interferes with action at the vasopressin receptors. Most commonly VRAs are used in the treatment... 10 KB (1,057 words) - 22:03, 12 March 2024 |
A receptor antagonist is a type of receptor ligand or drug that blocks or dampens a biological response by binding to and blocking a receptor rather than... 33 KB (3,837 words) - 09:01, 15 March 2024 |
boost the efficacy of 5-HT3 antagonists to prevent nausea and vomiting. The discovery of neurokinin 1 (NK1) receptor antagonists was a turning point in the... 29 KB (3,270 words) - 03:23, 5 December 2023 |
5-Hydroxytryptamine receptor 2B (5-HT2B) also known as serotonin receptor 2B is a protein that in humans is encoded by the HTR2B gene. 5-HT2B is a member... 33 KB (3,702 words) - 20:20, 16 April 2024 |
Mirtazapine (category Serotonin receptor antagonists) is not clear, but it may involve blocking certain adrenergic and serotonin receptors. Chemically, it is a tetracyclic antidepressant, and is closely related... 87 KB (7,798 words) - 22:33, 9 May 2024 |
Cariprazine (category Serotonin receptor antagonists) and D2 receptor partial agonist, with a preference for the D3 receptor. Cariprazine is also a partial agonist at the serotonin 5-HT1A receptor and acts... 30 KB (2,582 words) - 11:25, 27 April 2024 |
A cannabinoid receptor antagonist, also known simply as a cannabinoid antagonist or as an anticannabinoid, is a type of cannabinoidergic drug that binds... 41 KB (4,216 words) - 01:57, 28 March 2024 |
Anticholinergic (redirect from Acetylcholine receptor antagonist) anticholinergics by activating nicotinic acetylcholine receptors. Caffeine (although an adenosine receptor antagonist) can counteract the anticholinergic symptoms... 25 KB (2,388 words) - 23:35, 7 April 2024 |
Antihistamine (redirect from H1 receptor antagonist) receptor and heightens the receptor's activity; the receptor antagonists work by binding to the receptor and blocking the activation of the receptor by... 32 KB (3,138 words) - 14:01, 8 April 2024 |
An adenosine receptor antagonist is a drug which acts as an antagonist of one or more of the adenosine receptors. The best known are xanthines and their... 5 KB (458 words) - 09:41, 10 January 2024 |
Terguride (category Serotonin receptor antagonists) Accepted Name), sold under the brand name Teluron, is a serotonin receptor antagonist and dopamine receptor agonist of the ergoline family. It is approved for... 10 KB (526 words) - 14:46, 25 August 2023 |
Lisuride (category Serotonin receptor antagonists) as a mixed agonist and antagonist of dopamine, serotonin, and adrenergic receptors. Activation of specific dopamine receptors is thought to be responsible... 27 KB (2,067 words) - 03:25, 31 January 2024 |
Hydroxyzine (category Serotonin receptor antagonists) to act more weakly as an antagonist of the serotonin 5-HT2A receptor, the dopamine D2 receptor, and the α1-adrenergic receptor. Similarly to the atypical... 43 KB (3,708 words) - 17:28, 19 April 2024 |