The actions of vasopressin are mediated by stimulation of tissue-specific G protein-coupled receptors (GPCRs) called vasopressin receptors that are classified...
11 KB (974 words) - 03:10, 10 March 2024
Vasopressin receptor 1A (V1AR), or arginine vasopressin receptor 1A (officially called AVPR1A) is one of the three major receptor types for vasopressin...
29 KB (3,516 words) - 19:46, 7 January 2024
Vasopressin receptor 2 (V2R), or arginine vasopressin receptor 2 (officially called AVPR2), is a protein that acts as receptor for vasopressin. AVPR2 belongs...
15 KB (1,740 words) - 11:59, 4 January 2024
A vasopressin receptor antagonist (VRA) is an agent that interferes with action at the vasopressin receptors. Most commonly VRAs are used in the treatment...
10 KB (1,057 words) - 22:03, 12 March 2024
Human vasopressin, also called antidiuretic hormone (ADH), arginine vasopressin (AVP) or argipressin, is a hormone synthesized from the AVP gene as a...
43 KB (3,871 words) - 10:12, 24 March 2024
Vasopressin V1b receptor (V1BR) also known as vasopressin 3 receptor (VPR3) or antidiuretic hormone receptor 1B is a protein that in humans is encoded...
15 KB (1,757 words) - 03:12, 10 March 2024
vasopressin receptors TC OT 39 – non-selective over vasopressin receptors WAY-267,464 – anxiolytic in mice; possibly non-selective over vasopressin receptors...
22 KB (2,492 words) - 08:21, 9 May 2024
and V2 receptors which consequently lead to higher eGFR and lower vascular resistance in the lungs. A number of injectable arginine vasopressins are in...
25 KB (2,496 words) - 15:39, 20 December 2023
the vasopressin receptor 2 at the kidney (the site of ADH action); or inherited mutations leading to a gain of function of the vasopressin-2 receptor (a...
35 KB (4,043 words) - 10:29, 19 May 2024
AVP gene (section Vasopressin)
The arginine vasopressin gene (AVP) is a gene whose product is proteolytically cleaved to produce vasopressin (also known as antidiuretic hormone or ADH)...
21 KB (2,611 words) - 13:33, 12 March 2024
Desmopressin (redirect from 1-desamino-8-D-arginine vasopressin)
arterial hypertension. Vasopressin stimulates the release of ACTH, which indirectly increases responsiveness of alpha-1 receptor in blood vessel smooth...
17 KB (1,518 words) - 18:20, 7 November 2023
Oxytocin (category Vasopressin receptor agonists)
may be mediated by modulation of a different target, perhaps the vasopressin V1A receptor where oxytocin is known to weakly bind as an agonist. Oxytocin...
104 KB (11,642 words) - 16:05, 18 May 2024
Conivaptan (category Vasopressin receptor antagonists)
Vaprisol, is a non-peptide inhibitor of the receptor for anti-diuretic hormone, also called vasopressin. It was approved in 2004 for hyponatremia (low...
8 KB (805 words) - 10:03, 9 December 2022
(orexin) receptor 2 (HCRTR2, OX2R) Vasopressin receptor InterPro: IPR001817 Arginine vasopressin receptor 1A (AVPR1A, V1AR) Arginine vasopressin receptor 1B...
25 KB (2,172 words) - 01:01, 29 November 2023
Tolvaptan and conivaptan antagonize the effects of antidiuretic hormone (vasopressin), thereby promoting the specific excretion of free water, directly ameliorating...
38 KB (4,928 words) - 23:21, 28 December 2023
LIT-001 (category Vasopressin receptor agonists)
LIT-001 is a small-molecule oxytocin receptor agonist and vasopressin receptor mixed agonist and antagonist that was first described in the literature...
8 KB (691 words) - 17:41, 5 July 2023
Dopamine antagonist (redirect from Dopamine receptor antagonist)
anti-dopaminergic and a dopamine receptor antagonist (DRA), is a type of drug which blocks dopamine receptors by receptor antagonism. Most antipsychotics...
31 KB (3,140 words) - 02:58, 26 March 2024
not being produced in sufficient amounts, or vasopressin's receptors are not being stimulated by vasopressin. An example of desmopressin's use is for childhood...
3 KB (207 words) - 05:24, 9 September 2023
Nephrogenic diabetes insipidus (redirect from Arginine vasopressin resistance)
Nephrogenic diabetes insipidus, recently renamed as arginine vasopressin resistance (AVP-R) and also previously known as renal diabetes insipidus, is...
11 KB (1,191 words) - 18:38, 13 March 2024
Antihistamine (redirect from H1 receptor antagonist)
receptor and heightens the receptor's activity; the receptor antagonists work by binding to the receptor and blocking the activation of the receptor by...
32 KB (3,138 words) - 14:01, 8 April 2024
are not generally recommended. There is tentative evidence that vasopressin receptor antagonists (vaptans), such as conivaptan, may be slightly more effective...
39 KB (4,313 words) - 10:55, 9 May 2024
Tolvaptan (category Vasopressin receptor antagonists)
is an aquaretic drug that functions as a selective, competitive vasopressin receptor 2 (V2) antagonist used to treat hyponatremia (low blood sodium levels)...
11 KB (763 words) - 08:44, 15 May 2024
Terlipressin (category Vasopressin receptor agonists)
be effective when norepinephrine does not help. Terlipressin is a vasopressin receptor agonist. Terlipressin was approved for medical use in the United...
10 KB (584 words) - 08:21, 8 March 2024
S.; Orlandi, Cesare (2006-11-16). "Tolvaptan, a Selective Oral Vasopressin V2-Receptor Antagonist, for Hyponatremia". New England Journal of Medicine...
23 KB (1,998 words) - 12:42, 28 February 2024
adrenergic nerve synapses. Blockage of AT1 receptors directly causes vasodilation, reduces secretion of vasopressin, and reduces production and secretion of...
52 KB (5,143 words) - 12:34, 14 April 2024
Oxytocin (medication) (category Vasopressin receptor agonists)
oxytocin receptor agonists, like TC OT 39, WAY-267464, and LIT-001 have been developed and studied. However, lack of selectivity over vasopressin receptors has...
34 KB (3,243 words) - 19:40, 29 April 2024
Pharmacology (section Systems, receptors and ligands)
broad terms, pharmacodynamics discusses the chemicals with biological receptors, and pharmacokinetics discusses the absorption, distribution, metabolism...
48 KB (4,743 words) - 16:19, 27 April 2024
Dopaminergic (section Receptor agonists)
dopamine receptors can be classified as dopaminergic, and neurons that synthesize or contain dopamine and synapses with dopamine receptors in them may...
11 KB (1,161 words) - 01:41, 13 May 2024
Osmotherapy (section Vasopressin receptor antagonist)
glyburide (glibenclamide) which inhibits these channels. Vasopressin receptors activated by vasopressin are found on the basolateral membrane of the cells lining...
17 KB (2,050 words) - 06:15, 27 December 2023
Balovaptan (category Vasopressin receptor antagonists)
name RG7314), is a selective small molecule antagonist of the vasopressin V1A receptor which is under development by Roche for the treatment of post-traumatic...
6 KB (363 words) - 07:00, 21 April 2024